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Poly [ADP-ribose] polymerase 15 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
4,4'-OxydibenzamideIC504170.0 [1], 10000.0 [2]
OlaparibIC5017782.79 [1]
N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamideIC508912.51 [1]
RucaparibIC5032359.37 [1]
NiraparibIC5028840.32 [1]
Bmn-673 8R,9SIC5047863.01 [1]
4-MethoxybenzamideIC5010000.0 [1]
4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)-IC5017000.0 [1]
2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-oneIC5010000.0 [1]
2-[4-[6-[(3R,5S)-3,5-Dimethylpiperazin-1-yl]-4-methylpyridin-3-yl]phenyl]-7-methyl-3H-pyrrolo[2,3-d]pyrimidin-4-oneIC5025703.96 [1]
3-[[(Z)-4-[4-(4-Fluorophenyl)piperazin-1-yl]-4-oxobut-2-enoyl]amino]benzamideIC50520.0 [1]
(2z)-4-[(3-Carbamoylphenyl)amino]-4-Oxobut-2-Enoic AcidIC5015848.93 [1]
4-(4-Carbamoylphenoxy)benzoic acidIC502600.0 [1]
(2E)-4-[(3-Carbamoylphenyl)amino]-4-oxobut-2-enoic acidIC5017782.79 [1]
N-(3-Carbamoyl-phenyl)-succinamic acidIC5016218.1 [1]
4-[(2-Fluorophenyl)methoxy]benzamideIC503300.0 [1]
N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-MethoxybenzamideIC5010000.0 [1]
(Z)-4-(3-Carbamoylanilino)-3-methyl-4-oxobut-2-enoic acidIC5020000.0 [1]
(Z)-4-(3-Carbamoylanilino)-2-methyl-4-oxobut-2-enoic acidIC502344.23 [1]
2-[(3-Carbamoylphenyl)carbamoyl]cyclopentene-1-carboxylic acidIC501621.81 [1]
3-(3,4-Dimethyl-2,5-dioxopyrrol-1-yl)benzamideIC5010964.78 [1]
(Z)-N'-(3-Carbamoylphenyl)-N-methylbut-2-enediamideIC5020000.0 [1]
(E)-N'-(3-Carbamoylphenyl)-N-methylbut-2-enediamideIC5020000.0 [1]
3-[[(Z)-4-Oxo-4-pyrrolidin-1-ylbut-2-enoyl]amino]benzamideIC5016982.44 [1]
(Z)-N-(3-Carbamoylphenyl)-N',N'-diethylbut-2-enediamideIC5020000.0 [1]
Methyl (Z)-4-(3-carbamoylanilino)-4-oxobut-2-enoateIC501737.8 [1]
3-[(3-Oxocyclopentanecarbonyl)amino]benzamideIC5017782.79 [1]
1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrileIC5010000.0 [1]
2-(4-((Pyridin-4-Yl)methyl)piperazin-1-Yl)-3,4,5,6,7,8-Hexahydroquinazolin-4-OneIC5010000.0 [1]
4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC50100000.0 [1]
4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC50100000.0 [1]
5-(3-Carbamoylanilino)-5-oxopentanoic acidIC5020000.0 [1]
4-(4-Formyl-phenoxy)-benzamideIC5010000.0 [1]
1,2-Dihydro-2-(4-isopropylphenyl)-4(3H)-quinazolinoneIC5010000.0 [1]
3-(4-Oxopentanoylamino)benzamideIC5020000.0 [1]
2-[(3-Carbamoylphenyl)carbamoyl]cyclopropane-1-carboxylic acidIC5020000.0 [1]
4-(3-Carbamoylanilino)-2,2-dimethyl-4-oxobutanoic acidIC5020000.0 [1]
N-[3-Chloranyl-4-[[4-(4-Methoxyphenyl)oxan-4-Yl]methylcarbamoyl]phenyl]furan-2-CarboxamideIC5010000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Poly [ADP-ribose] polymerase 15 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-15-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Poly [ADP-ribose] polymerase 15 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-15-inhibitors-ic50-ki.
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