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Poly [ADP-ribose] polymerase 3 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
OlaparibIC5046.0 [1], 230.0 [2], 320.0 [3]
3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-oneIC50831.76 [1], 10000.0 [2]
NiraparibIC50296.0 [1], 1300.0 [2]
N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamideIC501430.0 [1]
VeliparibIC502040.0 [1]
RucaparibIC50512.0 [1]
Bmn-673 8R,9SIC5062.8 [1]
4-MethoxybenzamideIC50100000.0 [1]
3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-Phenylethyl]propanamideIC50900.0 [1]
4,4'-OxydibenzamideIC50100000.0 [1]
4-[[3-[(6S)-3-(1,1-Difluoroethyl)-6-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]-difluoromethyl]-2H-phthalazin-1-oneIC502800.0 [1]
5-(2-Oxo-2-phenylethoxy)isoquinolin-1(2H)-oneIC501300.0 [1]
4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)-IC5091000.0 [1]
2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-oneIC5034000.0 [1]
4-(4-Carbamoylphenoxy)benzoic acidIC50100000.0 [1]
4-[(2-Fluorophenyl)methoxy]benzamideIC50100000.0 [1]
2-[4-[3-[(4-Oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]pyridine-3-carbonitrileIC5046.0 [1]
N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-MethoxybenzamideIC50100000.0 [1]
1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrileIC50100000.0 [1]
PamiparibIC50185.0 [1]
3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-(Pyridin-2-Yl)ethyl]propanamideIC501300.0 [1]
3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1r)-1-(Pyridin-2-Yl)ethyl]propanamideIC50100000.0 [1]
3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-Phenylpropyl]propanamideIC502200.0 [1]
N-[(2s)-1-Hydroxy-3-Phenylpropan-2-Yl]-3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanamideIC501000.0 [1]
N-[(2s)-1-Hydroxybutan-2-Yl]-3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanamideIC509600.0 [1]
Methyl N-[3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanoyl]-L-PhenylalaninateIC502200.0 [1]
2-(4-((Pyridin-4-Yl)methyl)piperazin-1-Yl)-3,4,5,6,7,8-Hexahydroquinazolin-4-OneIC5013000.0 [1]
4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC5040000.0 [1]
4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC5045000.0 [1]
N-[1-(4-Imidazol-1-ylphenyl)ethyl]-3-(4-oxo-3H-quinazolin-2-yl)propanamideIC5013200.0 [1]
3-(4-Oxo-3,4-dihydroquinazolin-2-yl)-N-[1-(4-sulfamoylphenyl)ethyl]propanamideIC5014400.0 [1]
N-[(1R)-2,3-Dihydro-1H-inden-1-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamideIC50100000.0 [1]
N-[(1S)-2,3-Dihydro-1H-inden-1-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamideIC50100000.0 [1]
3-(4-Oxo-3H-quinazolin-2-yl)-N-[(1R)-1-phenylethyl]propanamideIC5015200.0 [1]
(2S)-2-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-3-phenylpropanamideIC503800.0 [1]
N-[(2S)-1-Hydroxypropan-2-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamideIC5011100.0 [1]
2-(3-Pyrazin-2-ylpropanoyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-oneIC5070.0 [1]
2-(2-Pyridin-3-ylacetyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-oneIC5050.0 [1]
4-(4-Formyl-phenoxy)-benzamideIC5086000.0 [1]
1,2-Dihydro-2-(4-isopropylphenyl)-4(3H)-quinazolinoneIC5050000.0 [1]
4-[(4s)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)benzamideIC5010000.0 [1]
7-(2-Fluorophenyl)-4-Methylquinolin-2(1h)-OneIC5010000.0 [1]
N-[3-Chloranyl-4-[[4-(4-Methoxyphenyl)oxan-4-Yl]methylcarbamoyl]phenyl]furan-2-CarboxamideIC50100000.0 [1]
6,7,16-Triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC50199.0 [1]
11-Fluoro-3,3-dimethyl-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC50136.0 [1]
3-Propan-2-yl-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC50760.0 [1]
3-(Cyclopropanecarbonyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC50180.0 [1]
3-(2,2-Dimethylpropanoyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC50660.0 [1]
3-(2-Amino-2-methylpropanoyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC5018.0 [1]
3,3-Dimethyl-16-(2-piperidin-1-ylethyl)-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC5020000.0 [1]
16-[2-(Diethylamino)ethyl]-3,3-dimethyl-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC5011000.0 [1]
3,3-Dimethyl-16-(oxiran-2-ylmethyl)-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-oneIC501000.0 [1]
4-[[4-Fluoro-3-[5-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]methyl]-2H-phthalazin-1-oneIC5066.9 [1]
Items per page: 1 - 10 of 53
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References

This online tool may be cited as follows

MLA

"Quest Database™ Poly [ADP-ribose] polymerase 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Poly [ADP-ribose] polymerase 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-3-inhibitors-ic50-ki.
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