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Poly [ADP-ribose] polymerase 4 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-oneIC504365.16 [1], 5011.87 [2]
NiraparibIC50330.0 [1], 446.68 [2]
OlaparibIC50407.38 [1]
N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamideIC50758.58 [1]
VeliparibIC503467.37 [1]
RucaparibIC50831.76 [1]
Bmn-673 8R,9SIC50257.04 [1]
4-MethoxybenzamideIC5065000.0 [1]
4,4'-OxydibenzamideIC5023000.0 [1]
4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)-IC5017000.0 [1]
Morpholin-4-Yl[4-(Tetrazolo[1,5-A]quinoxalin-4-Ylamino)phenyl]methanoneIC505011.87 [1]
2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-oneIC50100000.0 [1]
4-(4-Carbamoylphenoxy)benzoic acidIC50100000.0 [1]
4-[(2-Fluorophenyl)methoxy]benzamideIC50100000.0 [1]
N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-MethoxybenzamideIC50100000.0 [1]
1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrileIC50100000.0 [1]
2-(4-((Pyridin-4-Yl)methyl)piperazin-1-Yl)-3,4,5,6,7,8-Hexahydroquinazolin-4-OneIC5033000.0 [1]
4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC5069000.0 [1]
4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamideIC5065000.0 [1]
N-(4-Propan-2-ylphenyl)tetrazolo[1,5-a]quinoxalin-4-amineIC505011.87 [1]
2-(3-Pyrazin-2-ylpropanoyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-oneIC50660.0 [1]
2-(2-Pyridin-3-ylacetyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-oneIC50440.0 [1]
4-(4-Formyl-phenoxy)-benzamideIC50100000.0 [1]
1,2-Dihydro-2-(4-isopropylphenyl)-4(3H)-quinazolinoneIC50100000.0 [1]
[4-(1-Methylimidazole-4-carbonyl)piperazin-1-yl]-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanoneIC505011.87 [1]
(4-Pyrimidin-2-ylpiperazin-1-yl)-[4-(tetrazolo[1,5-a]quinoxalin-4-ylamino)phenyl]methanoneIC505011.87 [1]
N-[3-Chloranyl-4-[[4-(4-Methoxyphenyl)oxan-4-Yl]methylcarbamoyl]phenyl]furan-2-CarboxamideIC50100000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Poly [ADP-ribose] polymerase 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.10 May2024https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 10). Quest Database™ Poly [ADP-ribose] polymerase 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/poly-adp-ribose-polymerase-4-inhibitors-ic50-ki.
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