 | (3R,4S)-1-[(1S)-7-Fluoro-2,3-dihydro-1H-inden-1-yl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | IC50 | 290.0 [1], 660.0 [2] |
| (3R,4S)-1-[(1S)-7-Fluoro-2,3-dihydro-1H-inden-1-yl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | Ki | 1.0 [1], 11.0 [2] |
 | (3r,4s)-1-[(2-Bromo-6-Fluorophenyl)methyl]-N,N-Dimethyl-4-(1-Methyl-1h-Indol-3-Yl)pyrrolidin-3-Amine | IC50 | 4100.0 [1], 8300.0 [2] |
| (3r,4s)-1-[(2-Bromo-6-Fluorophenyl)methyl]-N,N-Dimethyl-4-(1-Methyl-1h-Indol-3-Yl)pyrrolidin-3-Amine | Ki | 10.0 [1], 13.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | IC50 | 2400.0 [1] |
| (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | Ki | 4.0 [1], 12.0 [2] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | IC50 | 33.0 [1], 50.0 [2] |
| 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 0.29 [1], 0.7 [2] |
 | 6-[4-[(3S,4R)-4-(Dimethylamino)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)pyrrolidin-3-yl]piperidin-1-yl]pyridine-3-carboxamide | IC50 | 230.0 [1], 280.0 [2] |
| 6-[4-[(3S,4R)-4-(Dimethylamino)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)pyrrolidin-3-yl]piperidin-1-yl]pyridine-3-carboxamide | Ki | 0.45 [1] |
 | 4-[3-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-1-methylindol-7-yl]-1-methylpiperazin-2-one | IC50 | 100.0 [1], 190.0 [2] |
| 4-[3-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-1-methylindol-7-yl]-1-methylpiperazin-2-one | Ki | 0.74 [1] |
 | [3-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-1-methylindol-7-yl]-(3-fluoroazetidin-1-yl)methanone | IC50 | 31.0 [1], 180.0 [2] |
| [3-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-1-methylindol-7-yl]-(3-fluoroazetidin-1-yl)methanone | Ki | 1.0 [1] |
 | (3R,4S)-1-[(2-Chloro-6-fluorophenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | IC50 | 6900.0 [1], 10000.0 [2] |
| (3R,4S)-1-[(2-Chloro-6-fluorophenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | Ki | 53.0 [1] |
 | (1S,2R)-4-(7-Fluoro-2,3-dihydro-1H-inden-1-yl)-N,N-dimethyl-2-[4-(4-methylsulfonylpiperazin-1-yl)phenyl]cyclopentan-1-amine | IC50 | 44.0 [1], 57.0 [2] |
| (1S,2R)-4-(7-Fluoro-2,3-dihydro-1H-inden-1-yl)-N,N-dimethyl-2-[4-(4-methylsulfonylpiperazin-1-yl)phenyl]cyclopentan-1-amine | Ki | 0.3 [1] |
 | 9-Benzyl-5-(furan-2-ylmethylamino)-8,10-dihydro-7H-[1,2,4]triazolo[3,4-a][2,7]naphthyridine-6-carbonitrile | IC50 | 620.0 [1], 3280.0 [2], 4030.0 [3] |
 | Tazemetostat | IC50 | 2.0 [1], 40.0 [2] |
 | N-(Furan-2-Ylmethyl)-8-(4-Methylsulfonylphenyl)-[1,2,4]triazolo[4,3-C]pyrimidin-5-Amine | IC50 | 22.0 [1], 220.0 [2] |
 | CID 123132213 | IC50 | 7.0 [1] |
| CID 123132213 | Ki | 0.3 [1] |
 | (3r,4s)-1-[(2-Methoxyphenyl)methyl]-N,N-Dimethyl-4-(1-Methylindol-3-Yl)pyrrolidin-3-Amine | Ki | 600.0 [1] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 2.6 [1], 3.0 [2] |
 | (3R,4S)-1-[(2-Bromo-6-fluorophenyl)methyl]-N,N-dimethyl-4-phenylpyrrolidin-3-amine | Ki | 78.0 [1], 110.0 [2] |
 | 1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-N,N-dimethylpiperidine-4-carboxamide | IC50 | 40.0 [1], 70.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-[4-(4-methylphenyl)piperazin-1-yl]phenyl]pyrrolidin-3-amine | IC50 | 150.0 [1], 220.0 [2] |
 | 1-[1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperidin-4-yl]pyrrolidin-2-one | IC50 | 80.0 [1], 120.0 [2] |
 | [4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylphenyl]-(4-ethylpiperazin-1-yl)methanone | IC50 | 290.0 [1], 460.0 [2] |
 | (3R,4S)-4-[4-(6,8-Dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)phenyl]-1-[(2-fluoro-6-methylphenyl)methyl]-N,N-dimethylpyrrolidin-3-amine | IC50 | 130.0 [1], 210.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-pyridin-3-ylbenzamide | IC50 | 80.0 [1], 100.0 [2] |
 | 1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-N-methylpiperidine-4-carboxamide | IC50 | 50.0 [1], 110.0 [2] |
 | 6-(1,3-Benzodioxol-4-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-3-amine | IC50 | 1000.0 [1], 1300.0 [2] |
 | 8-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one | IC50 | 60.0 [1], 140.0 [2] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylbenzoyl]piperazin-1-yl]ethanone | IC50 | 180.0 [1], 510.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-pyridin-4-ylbenzamide | IC50 | 80.0 [1], 90.0 [2] |
 | (3R,4S)-4-[4-(6,8-Dihydro-5H-imidazo[1,2-a]pyrazin-7-yl)phenyl]-1-[(2-fluoro-6-methylphenyl)methyl]-N,N-dimethylpyrrolidin-3-amine | IC50 | 70.0 [1], 100.0 [2] |
 | 4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-1-ethylpiperazin-2-one | IC50 | 60.0 [1], 120.0 [2] |
 | Methyl 4-[4-[(3S,4R)-4-(dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperazine-1-carboxylate | IC50 | 30.0 [1], 40.0 [2] |
 | N-[1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperidin-4-yl]acetamide | IC50 | 40.0 [1], 160.0 [2] |
 | Cyclopropyl-[4-[4-[(3S,4R)-4-(dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylbenzoyl]piperazin-1-yl]methanone | IC50 | 340.0 [1], 440.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-(4-phenylpiperazin-1-yl)phenyl]pyrrolidin-3-amine | IC50 | 50.0 [1], 90.0 [2] |
 | 1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-N,N-dimethylpiperidin-4-amine | IC50 | 40.0 [1], 100.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide | IC50 | 80.0 [1], 100.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-[4-(2-methylsulfonylphenyl)piperazin-1-yl]phenyl]pyrrolidin-3-amine | IC50 | 70.0 [1], 190.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-4-[4-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]phenyl]-N,N-dimethylpyrrolidin-3-amine | IC50 | 40.0 [1], 50.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-(pyridin-3-ylmethyl)benzamide | IC50 | 80.0 [1], 100.0 [2] |
 | N-[(3S)-1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]pyrrolidin-3-yl]acetamide | IC50 | 90.0 [1], 240.0 [2] |
 | 6-[(2-Fluoro-5-methoxyphenyl)methyl]-1-propan-2-yl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-3-amine | IC50 | 1300.0 [1], 2900.0 [2] |
 | 2-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-3,6,7,8,9,9a-hexahydro-1H-pyrido[1,2-a]pyrazin-4-one | IC50 | 100.0 [1], 170.0 [2] |
 | [4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylphenyl]-[4-(2-hydroxyethyl)piperazin-1-yl]methanone | IC50 | 270.0 [1], 380.0 [2] |
 | [4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylphenyl]-pyrrolidin-1-ylmethanone | IC50 | 140.0 [1], 260.0 [2] |
 | 4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-N,N-dimethylpiperazine-1-sulfonamide | IC50 | 20.0 [1], 60.0 [2] |
 | [4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylphenyl]-(4-methyl-1,4-diazepan-1-yl)methanone | IC50 | 310.0 [1], 390.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-N,N,2-trimethylbenzamide | IC50 | 110.0 [1], 180.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]phenyl]pyrrolidin-3-amine | IC50 | 50.0 [1], 80.0 [2] |
 | 3-(1-Benzofuran-7-ylmethyl)piperidine-1-carboximidamide | IC50 | 2500.0 [1], 2800.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-(pyridin-2-ylmethyl)benzamide | IC50 | 70.0 [1], 80.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-(4-pyridin-4-ylpiperazin-1-yl)phenyl]pyrrolidin-3-amine | IC50 | 10.0 [1] |
 | 6-(1-Benzofuran-4-ylmethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-3-amine | IC50 | 2700.0 [1], 12400.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-(pyridin-4-ylmethyl)benzamide | IC50 | 70.0 [1], 110.0 [2] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-1,4-diazepan-1-yl]ethanone | IC50 | 160.0 [1], 270.0 [2] |
 | (4-Chlorophenyl)-[4-[4-[(3S,4R)-4-(dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]methanone | IC50 | 20.0 [1], 40.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methyl-N-[2-(4-methylpiperazin-1-yl)ethyl]benzamide | IC50 | 90.0 [1], 120.0 [2] |
 | 8-(2-Fluorophenyl)-5-(furan-2-ylmethylamino)-[1,2,4]triazolo[4,3-a]pyridine-6-carbonitrile | IC50 | 30.0 [1], 210.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-(4-morpholin-4-ylpiperidin-1-yl)phenyl]pyrrolidin-3-amine | IC50 | 40.0 [1], 60.0 [2] |
 | 1-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperidine-4-carbonitrile | IC50 | 70.0 [1], 140.0 [2] |
 | [4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]-pyrrolidin-1-ylmethanone | IC50 | 30.0 [1], 40.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-(4-pyrimidin-2-ylpiperazin-1-yl)phenyl]pyrrolidin-3-amine | IC50 | 30.0 [1], 70.0 [2] |
 | 3-(1-Benzofuran-4-ylmethyl)piperidine-1-carboximidamide | IC50 | 2100.0 [1], 2500.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-N,N-diethyl-2-methylbenzamide | IC50 | 100.0 [1], 250.0 [2] |
 | 3-(1,3-Benzodioxol-4-ylmethyl)piperidine-1-carboximidamide | IC50 | 1600.0 [1], 3900.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-[4-(1,3-thiazol-2-yl)piperazin-1-yl]phenyl]pyrrolidin-3-amine | IC50 | 30.0 [1], 40.0 [2] |
 | [4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylphenyl]-(4-methylpiperazin-1-yl)methanone | IC50 | 260.0 [1], 480.0 [2] |
 | N-(Furan-2-ylmethyl)-8-[4-(pyrrolidin-1-ylmethyl)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine | IC50 | 7.0 [1], 32.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-N-(2-methoxyethyl)-N,2-dimethylbenzamide | IC50 | 130.0 [1], 140.0 [2] |
 | N-[2-(Dimethylamino)ethyl]-4-[(3S,4R)-4-(dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-2-methylbenzamide | IC50 | 80.0 [1], 150.0 [2] |
 | 4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]-N,2-dimethyl-N-(oxolan-2-ylmethyl)benzamide | IC50 | 110.0 [1], 290.0 [2] |
 | N-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]-N,1-dimethylpiperidin-4-amine | IC50 | 90.0 [1], 350.0 [2] |
 | 8-(1,3-Benzodioxol-4-ylmethyl)-1-propan-2-yl-5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-3-amine | IC50 | 430.0 [1], 2000.0 [2] |
 | (3R,4S)-1-[(2-Fluoro-6-methylphenyl)methyl]-N,N-dimethyl-4-[4-(4-methylpiperidin-1-yl)phenyl]pyrrolidin-3-amine | IC50 | 40.0 [1], 140.0 [2] |
 | Astemizole | IC50 | 93800.0 [1] |
 | 3-Benzylpiperidine | IC50 | 500000.0 [1] |
 | 5-(2-Fluoro-phenyl)-2,3-dihydro-imidazo[2,1-a]isoquinoline | IC50 | 6040.0 [1] |
 | 2-Pyridin-4-yl-1,2,3,4-tetrahydro-isoquinoline | Ki | 950.0 [1] |
 | 9-Benzyl-5-chloro-7,8,9,10-tetrahydro-[1,2,4]triazolo[3,4-a][2,7]naphthyridine-6-carbonitrile | IC50 | 100000.0 [1] |
 | [(5S)-6-[[(2S)-1-[[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-5-[[(2S)-3-hydroxy-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoyl]amino]-6-oxohexyl]-trimethylazanium | IC50 | 1650.0 [1] |
 | 2-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(2-fluoro-6-methylphenyl)methyl]pyrrolidin-3-yl]phenyl]pyrazol-1-yl]acetamide | Ki | 2.6 [1] |
 | (3R,4S)-1-[(1R)-7-Fluoro-2,3-dihydro-1H-inden-1-yl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | Ki | 129.0 [1] |
 | 1-[4-[4-[(3R,4S)-4-(Dimethylamino)-1-[(1R)-7-fluoro-2,3-dihydro-1H-inden-1-yl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 18.0 [1] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(1S)-7-fluoro-2,3-dihydro-1H-inden-1-yl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 0.3 [1] |
 | 1-[4-[4-[(3S,4R)-4-(Dimethylamino)-1-[(1R)-7-fluoro-2,3-dihydro-1H-inden-1-yl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 3.0 [1] |
 | 1-[4-[4-[(3R,4S)-4-(Dimethylamino)-1-[(1S)-7-fluoro-2,3-dihydro-1H-inden-1-yl]pyrrolidin-3-yl]phenyl]piperazin-1-yl]ethanone | Ki | 42.0 [1] |
 | (3R,4As,10aS)-6-methoxy-3-[(3-methoxyphenyl)methyl]-1-methyl-3,4,4a,5,10,10a-hexahydro-2H-benzo[g]quinoline | IC50 | 2500.0 [1] |
 | 5-(Furan-2-ylmethylamino)-[1,2,4]triazolo[4,3-a]pyridine-6-carbonitrile | IC50 | 1000.0 [1] |
 | 8-[4-[(Dimethylamino)methyl]phenyl]-N-[(3-methylthiophen-2-yl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine | IC50 | 49.0 [1] |
 | 8-[4-[(Dimethylamino)methyl]phenyl]-5-[(5-fluorothiophen-2-yl)methylamino]-[1,2,4]triazolo[4,3-a]pyridine-6-carbonitrile | IC50 | 510.0 [1] |
 | 5-(Furan-2-ylmethylamino)-8-phenyl-[1,2,4]triazolo[4,3-a]pyridine-6-carbonitrile | IC50 | 62.0 [1] |
 | (3S,4R)-1-[(2-Bromo-6-fluorophenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine | Ki | 80.0 [1] |
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