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Prostanoid EP1 receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
3-(2-(2-(Benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acidIC507.94 [1], 1.25892541179417e+17 [2]
3-(2-(2-(Benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acidKi0.71 [1]
3-(3-(2-(Benzyloxy)-5-chlorophenyl)thiophen-2-yl)benzoic acidIC503.55 [1], 5.0 [2]
3-(3-(2-(Benzyloxy)-5-chlorophenyl)thiophen-2-yl)benzoic acidKi0.3 [1], 1.26 [2], 4.0 [3], 70.0 [4]
2-(4-Methyl-3,5-diphenyl-1H-pyrazole-1-yl)-4-thiazolecarboxylic acidIC5050.0 [1], 500.0 [2]
2-(4-Methyl-3,5-diphenyl-1H-pyrazole-1-yl)-4-thiazolecarboxylic acidKi290.0 [1]
3-[2-(5-Chloro-2-phenylmethoxyphenyl)phenyl]benzoic acidIC5050.12 [1]
3-[2-(5-Chloro-2-phenylmethoxyphenyl)phenyl]benzoic acidKi28.84 [1], 31.62 [2]
DinoprostoneIC501.1 [1]
DinoprostoneKi9.1 [1], 18.0 [2]
2-Pyridinecarboxylic acid, 6-(5'-chloro-2'-(2-methylpropoxy)(1,1'-biphenyl)-2-yl)-, sodium saltIC5015.85 [1], 16.0 [2]
2-Pyridinecarboxylic acid, 6-(5'-chloro-2'-(2-methylpropoxy)(1,1'-biphenyl)-2-yl)-, sodium saltKi2.51 [1]
3-(2-(2-(Benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)benzoic acidIC505.01 [1], 12.59 [2]
3-(2-(2-(Benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)benzoic acidKi4.27 [1]
2-(6-Trifluoromethyl-3-phenyl-1H-indazole-1-yl)-4-thiazolecarboxylic acidIC500.6 [1], 14.0 [2]
2-(6-Trifluoromethyl-3-phenyl-1H-indazole-1-yl)-4-thiazolecarboxylic acidKi0.45 [1]
6-[2-[5-Chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-1-cyclopentenyl]pyridine-2-carboxylic AcidIC502.51 [1]
Acetic acid, (3-(((1S)-2-(4,5-diphenyl-2-oxazolyl)-2-cyclohexen-1-yl)methyl)phenoxy)-, sodium saltKi1000.0 [1]
3-(2-(2-(4-Fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acidIC506.31 [1]
2-{2-Ethyl[(4-methylphenyl)sulfonyl]anilino}-N-(4-methoxybenzyl)acetamideIC5025.0 [1]
2-{2-Ethyl[(4-methylphenyl)sulfonyl]anilino}-N-(4-methoxybenzyl)acetamideKi25.12 [1], 35.48 [2]
3-(2-(2-(Benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acidIC5010.0 [1]
3-(2-(2-(Benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acidKi0.59 [1]
1-(2-(Benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acidIC506.31 [1], 6.46 [2]
1-(2-(Benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acidKi15.14 [1]
2-(4-Amino-3,5-diphenyl-1H-pyrazole-1-yl)-4-thiazolecarboxylic acidIC5020.0 [1], 60.0 [2]
2-(4-Amino-3,5-diphenyl-1H-pyrazole-1-yl)-4-thiazolecarboxylic acidKi8.0 [1]
2-[5-(4-Methoxyphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carboxylic acidIC501000.0 [1], 5800.0 [2]
2-[5-(4-Methoxyphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carboxylic acidKi8700.0 [1]
2-[3-(2-Hydroxyphenyl)-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carboxylic acidIC50180.0 [1], 800.0 [2]
2-[3-(2-Hydroxyphenyl)-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carboxylic acidKi530.0 [1]
DinoprostIC50220.0 [1], 380.0 [2]
1-[5-[3-(5-Chloro-2-phenylmethoxyphenyl)thiophen-2-yl]pyridin-3-yl]-2,2,2-trifluoroethane-1,1-diolKi4.0 [1], 5.0 [2]
2-[(3R)-5-Acetyl-4-[(4-chlorophenyl)methyl]-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidKi20000.0 [1]
Sodium 6-((5-chloro-2-(((4-chloro-2-fluorophenyl)methyl)oxy)phenyl)methyl)-2-pyridinecarboxylateIC5012.59 [1]
Sodium 6-((5-chloro-2-(((4-chloro-2-fluorophenyl)methyl)oxy)phenyl)methyl)-2-pyridinecarboxylateKi7.94 [1]
N-[2-(4-Chlorophenyl)ethyl]-2-(2-methyl-N-(4-methylphenyl)sulfonylanilino)acetamideIC50251.19 [1]
N-[2-(4-Chlorophenyl)ethyl]-2-(2-methyl-N-(4-methylphenyl)sulfonylanilino)acetamideKi660.69 [1]
(E)-3-{2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acidKi12000.0 [1]
(E)-3-[2-(3,4-Dichlorophenyl)phenyl]-N-thiophen-2-ylsulfonylprop-2-enamideKi8100.0 [1], 8200.0 [2]
3-[2-[5-Chloro-2-(2-methylpropoxy)phenyl]-5-methylpyrrol-1-yl]benzoic acidIC505.01 [1]
2-[(3R)-4-[(4-Chlorophenyl)methyl]-5-(1-hydroxyethyl)-7-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acidKi20000.0 [1]
2-(2-Benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acidIC5010000.0 [1], 25000.0 [2]
7-{(R)-2-[(E)-3-Hydroxy-3-(1-phenyl-cyclopropyl)-propenyl]-5-oxo-pyrrolidin-1-yl}-heptanoic acidKi13000.0 [1], 28000.0 [2]
7-[3,5-Dihydroxy-2-(3-hydroxy-5-phenyl-pentyl)-cyclopentyl]-heptanoic acidIC501100.0 [1], 5600.0 [2]
5-(2-(2-(Benzyloxy)-5-(trifluoromethyl)phenyl)cyclopent-1-enyl)nicotinic acidIC5010.0 [1]
3-(2-((E)-3-(4-(Benzyloxy)-3-methoxyphenyl)prop-1-enyl)phenyl)-N-(thiophen-2-ylsulfonyl)acrylamideKi1500.0 [1], 2443.0 [2]
N-[2-(3,4-Dimethoxyphenyl)ethyl]-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamideIC507.94 [1]
N-[2-(3,4-Dimethoxyphenyl)ethyl]-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamideKi13.49 [1]
Sodium;2-(5-chloro-2-phenylmethoxyanilino)-1,3-thiazole-4-carboxylateIC5025.12 [1]
Sodium;2-[[5-chloro-2-(2-methylpropoxy)phenyl]methyl]-1,3-thiazole-4-carboxylateIC507.94 [1]
Sodium;6-[[5-chloro-2-(2-methylpropoxy)phenyl]methyl]pyridine-2-carboxylateIC5039.81 [1]
N-[5-(2,6-Dichlorophenyl)-1,3,4-thiadiazol-2-yl]-4-ethyl-2,3-dihydro-1,4-benzoxazine-6-carboxamideKi10000.0 [1], 25118.86 [2]
3-(2-(2-(Benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acidIC507.94 [1]
4-[2-(5-Chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamideIC502.51 [1], 3.98107170553499e+17 [2]
N-Benzyl-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamideIC5025.12 [1], 3.98107170553499e+16 [2]
N-[1-[(5-Chloro-2-phenylmethoxyphenyl)methyl]-5-methylpyrazol-3-yl]benzamideIC5015.85 [1], 6.30957344480194e+16 [2]
1-[(5-Chloro-2-phenylmethoxyphenyl)methyl]-5-methyl-N-phenylpyrazole-3-carboxamideIC5039.81 [1], 2.51188643150957e+16 [2]
Sodium;1-[(5-bromo-2-phenylmethoxyphenyl)methyl]-5-methylpyrazole-3-carboxylateIC506.31 [1], 1.58489319246111e+17 [2]
Sodium;6-[(5-chloro-2-phenylmethoxyphenyl)methyl]pyridine-2-carboxylateIC50158.49 [1]
Sodium;1-[(5-chloro-2-phenylmethoxyphenyl)methyl]-5-methylpyrazole-3-carboxylateIC5010.0 [1]
(E)-3-[2-[(E)-3-Phenylprop-1-enyl]phenyl]prop-2-enoic acid;(E)-3-[2-[(E)-3-phenylprop-2-enyl]phenyl]prop-2-enoic acidKi100000.0 [1]
(E)-3-[2-[(E)-3-(4-Methoxyphenyl)prop-1-enyl]phenyl]prop-2-enoic acid;(E)-3-[2-[(E)-3-(4-methoxyphenyl)prop-2-enyl]phenyl]prop-2-enoic acidKi100000.0 [1]
3-(2-(Naphthalen-2-ylmethyl)phenyl)acrylic acidKi100000.0 [1]
N-Benzyl-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamideKi63.1 [1], 223.87 [2]
3-Acetamido-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acidIC500.4 [1]
3-Acetamido-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acidKi0.1 [1]
3-(5-(2-(Benzyloxy)-5-chlorophenyl)-1H-imidazol-1-yl)benzoic acidIC50125.89 [1]
3-(5-(2-(Benzyloxy)-5-chlorophenyl)-1H-imidazol-1-yl)benzoic acidKi3.55 [1]
5-[2-[5-Chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acidIC505.01 [1]
5-[2-[5-Chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acidKi1.0 [1]
1-{5-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-pyridin-3-yl}-2,2,2-trifluoro-ethanolKi3.0 [1], 6.0 [2]
1-[[5-Bromo-2-[(4-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC508.71 [1]
1-[[5-Bromo-2-[(4-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi8.71 [1]
1-[[5-Bromo-2-[(2-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC503.16 [1]
1-[[5-Bromo-2-[(2-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi28.84 [1]
1-[(5-Bromo-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)methyl]-5-methyl-1H-pyrazole-3-carboxylic acidIC500.52 [1]
1-[(5-Bromo-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)methyl]-5-methyl-1H-pyrazole-3-carboxylic acidKi2.63 [1]
3-(3-(2-(Benzyloxy)-5-chlorophenyl)pyridin-2-yl)benzoic acidIC50100.0 [1]
3-(3-(2-(Benzyloxy)-5-chlorophenyl)pyridin-2-yl)benzoic acidKi6.61 [1]
1-[[2-[(2,4-Dichlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC501995.26 [1]
1-[[2-[(2,4-Dichlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi8.32 [1]
1-[[5-Bromo-2-[(3-methylphenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC50125.89 [1]
1-[[5-Bromo-2-[(3-methylphenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi524.81 [1]
1-[[5-Bromo-2-[(3-bromophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC5017.78 [1]
1-[[5-Bromo-2-[(3-bromophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi128.82 [1]
1-[[2-[(2,4-Dichlorophenyl)methoxy]-5-fluorophenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC50354.81 [1]
1-[[2-[(2,4-Dichlorophenyl)methoxy]-5-fluorophenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi20.42 [1]
1-[[5-Bromo-2-[(3-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC50114.82 [1]
1-[[5-Bromo-2-[(3-chlorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidKi426.58 [1]
1-[(5-Bromo-2-phenylmethoxyphenyl)methyl]-5-thiophen-2-ylpyrazole-3-carboxylic acidIC50194.98 [1]
1-[(5-Bromo-2-phenylmethoxyphenyl)methyl]-5-thiophen-2-ylpyrazole-3-carboxylic acidKi616.6 [1]
EP1-antagonist-1IC500.13 [1]
EP1-antagonist-1Ki0.49 [1]
3-[4-(5-Chloro-2-phenylmethoxyphenyl)pyridin-3-yl]benzoic acidIC50316.23 [1]
3-[4-(5-Chloro-2-phenylmethoxyphenyl)pyridin-3-yl]benzoic acidKi28.18 [1]
1-[(5-Bromo-2-phenylmethoxyphenyl)methyl]pyrazole-3-carboxylic acidIC509.77 [1]
1-[(5-Bromo-2-phenylmethoxyphenyl)methyl]pyrazole-3-carboxylic acidKi54.95 [1]
3-[2-(5-Chloro-2-phenylmethoxyphenyl)thiophen-3-yl]benzenesulfonamideKi8.0 [1], 18.0 [2]
1-[[5-Chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]methyl]-5-methylpyrazole-3-carboxylic acidIC501995.26 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Prostanoid EP1 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/prostanoid-ep1-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Prostanoid EP1 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/prostanoid-ep1-receptor-inhibitors-ic50-ki.
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