logo
Products
Technologies
Applications
Services
Resources
Selection Guides
About
Prostanoid EP4 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
DinoprostoneIC500.7 [1]
DinoprostoneKi0.79 [1], 3.1 [2]
GrapiprantIC5011.7 [1]
GrapiprantKi13.0 [1], 448.0 [2], 449.0 [3]
1-(2,6-Dichlorophenyl)sulfonyl-3-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]ureaIC503.0 [1], 14.0 [2], 78.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseProstanoid EP4 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.31 Dec2025https://www.aatbio.com/data-sets/prostanoid-ep4-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 31). Quest DatabaseProstanoid EP4 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/prostanoid-ep4-receptor-inhibitors-ic50-ki.
BibTeXEndNoteRefMan