Prostasin Inhibitors (IC50, Ki)

Name: Prostasin Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[(4-chlorophenyl)methoxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	12.0 ^[1]
	Benzyl N-[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamate	Ki	100000.0 ^[1]
	Benzyl N-[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	100000.0 ^[1]
	Benzyl N-[(2S)-6-amino-1-[[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]carbamate	Ki	15200.0 ^[1]
	Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamate	Ki	5720.0 ^[1]
	Benzyl N-[(2S)-6-amino-1-[[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]amino]-1-oxohexan-2-yl]carbamate	Ki	5780.0 ^[1]
	Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamate	Ki	2100.0 ^[1]
	Benzyl N-[(2R)-1-[(2S)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	1400.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,3R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-3-phenylpyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	267.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,3S)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-3-methylpyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	49.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-phenylmethoxypyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	40.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	1040.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[[3-(trifluoromethyl)phenyl]methoxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	41.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[[4-(trifluoromethyl)phenyl]methoxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	28.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[(4-methylphenyl)methoxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	45.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[(4-fluorophenyl)methoxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	27.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-(cyclohexylmethoxy)pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	19.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-(cyclopentylmethoxy)pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	65.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-(phenylcarbamoyloxy)pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	130.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-(benzylcarbamoyloxy)pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	60.0 ^[1]
	Benzyl N-[(2R)-1-[(2S,4R)-2-[[(2S)-6-amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-4-[(4-methylsulfonylphenyl)methylcarbamoyloxy]pyrrolidin-1-yl]-1-oxo-4-phenylbutan-2-yl]carbamate	Ki	176.0 ^[1]
	[(3R,5S)-5-[[(2S)-6-Amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-1-[(2R)-4-phenyl-2-(phenylmethoxycarbonylamino)butanoyl]pyrrolidin-3-yl] piperidine-1-carboxylate	Ki	29.0 ^[1]
	[(3R,5S)-5-[[(2S)-6-Amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-1-[(2R)-4-phenyl-2-(phenylmethoxycarbonylamino)butanoyl]pyrrolidin-3-yl] pyrrolidine-1-carboxylate	Ki	101.0 ^[1]
	[(3R,5S)-5-[[(2S)-6-Amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-1-[(2R)-4-phenyl-2-(phenylmethoxycarbonylamino)butanoyl]pyrrolidin-3-yl] morpholine-4-carboxylate	Ki	510.0 ^[1]
	[(3R,5S)-5-[[(2S)-6-Amino-1-(1,3-benzoxazol-2-yl)-1-oxohexan-2-yl]carbamoyl]-1-[(2R)-4-phenyl-2-(phenylmethoxycarbonylamino)butanoyl]pyrrolidin-3-yl] N,N-dimethylcarbamate	Ki	1550.0 ^[1]

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References

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MLA	"Quest Database™ Prostasin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/prostasin-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Prostasin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/prostasin-inhibitors-ic50-ki.
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Prostasin Inhibitors (IC50, Ki)

References

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MLA

APA