Products
Technologies
Applications
Services
Resources
Selection Guides
About
Proteasome Macropain subunit Inhibitors (IC50, Ki)
Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
 | Bortezomib | IC50 | 1880.0 [1] |
 | Z-Leu-leu-leu-al | IC50 | 52.0 [1], 2100.0 [2] |
| Z-Leu-leu-leu-al | Ki | 1.0 [1], 330.0 [2], 5520.0 [3], 22100.0 [4] |
 | (2S)-N-[(2S)-1-[[(E,2S)-1-[4-(Aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-4-methylpentanamide | IC50 | 10.8 [1], 50.0 [2], 84.0 [3], 170.0 [4], 2700.0 [5] |
 | (2S)-N-[(E,2S)-1-[4-(Aminomethyl)phenyl]-4-methylsulfonylbut-3-en-2-yl]-2-[[(2S)-3-(4-aminophenyl)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanamide | IC50 | 47.0 [1], 110.0 [2], 580.0 [3], 10000.0 [4] |
References
This online resource may be cited as follows
MLA | "Quest Database™ Proteasome Macropain subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 Dec. 2025, https://www.aatbio.com/data-sets/proteasome-macropain-subunit-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 8). Quest Database™ Proteasome Macropain subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/proteasome-macropain-subunit-inhibitors-ic50-ki. | |
| BibTeX | EndNote | RefMan |