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Proteasome Macropain subunit MB1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
BortezomibIC504.68 [1]
BortezomibKi0.55 [1], 0.6 [2], 9.8 [3]
Z-Leu-leu-leu-alIC509.0 [1], 11.0 [2], 25.0 [3], 37.0 [4]
Z-Leu-leu-leu-alKi1.4 [1], 3.7 [2], 4.0 [3], 70.0 [4]
5-Aminoquinolin-8-olIC50600.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseProteasome Macropain subunit MB1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/proteasome-macropain-subunit-mb1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseProteasome Macropain subunit MB1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/proteasome-macropain-subunit-mb1-inhibitors-ic50-ki.
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