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Protein AF-9 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-3-amino-1-[[(2S)-3-cyclopentyl-1-[(2S)-2-(1-methyl-4-phenylimidazol-2-yl)pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi57.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-3-amino-1-[[(2S)-1-[(2S)-2-[1-(cyclohexylmethyl)-4-phenylimidazol-2-yl]pyrrolidin-1-yl]-3-cyclopentyl-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi13.0 [1]
(2S)-N-[(2S)-1-[[(2S)-3-Amino-1-[[(2S)-1-[(2S)-2-[1-(cyclohexylmethyl)-4-phenylimidazol-2-yl]pyrrolidin-1-yl]-3-cyclopentyl-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-1-(4-methylpentanoyl)pyrrolidine-2-carboxamideKi23.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-cyclopentylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi130.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-3-amino-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi190.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-naphthalen-2-ylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi730.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi170.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(1S)-1-cyclopentyl-2-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-2-oxoethyl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi250.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi20.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-3-cyclobutyl-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]pyrrolidine-2-carboxamideKi1310.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-phenylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi280.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-naphthalen-1-ylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi2600.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamideKi5620.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-3-amino-1-[[(2S)-3-cyclopentyl-1-[(2S)-2-(1-ethyl-4-phenylimidazol-2-yl)pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi50.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-3-amino-1-[[(2S)-3-cyclopentyl-1-oxo-1-[(2S)-2-(4-phenyl-1-propan-2-ylimidazol-2-yl)pyrrolidin-1-yl]propan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi57.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-3-cyclopropyl-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]pyrrolidine-2-carboxamideKi780.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi300.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-aminopropanoyl]amino]-3-cyclopentylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi20.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi830.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi410.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-cyclohexylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi180.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[6-[5-[(3Ar,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-aminopropanoyl]amino]-3-cyclopentylpropanoyl]-N-[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi10.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(1S)-1-cyclohexyl-2-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-2-oxoethyl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi620.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi160.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S,3S)-1-[[(2S)-5-amino-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi4250.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-(dimethylamino)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideKi1160.0 [1]
(2S)-1-[(2S)-2-Acetamido-4-methylpentanoyl]-N-[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[(2S)-2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]pyrrolidine-2-carboxamideKi160.0 [1]
(2S)-N-[(2S)-1-[[(2S)-3-Amino-1-[[(2S)-1-[(2S)-2-[1-(cyclohexylmethyl)-4-phenylimidazol-2-yl]pyrrolidin-1-yl]-3-cyclopentyl-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-1-benzoylpyrrolidine-2-carboxamideKi9.0 [1]
Items per page: 1 - 10 of 28
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein AF-9 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/protein-af-9-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Protein AF-9 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-af-9-inhibitors-ic50-ki.
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