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Protein-arginine deiminase type-4 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Cl-amidine (TFA)IC503400.0 [1], 4000.0 [2], 9000.0 [3], 15000.0 [4]
Cl-amidine (TFA)Ki180000.0 [1]
F-AmidineIC5015000.0 [1], 21000.0 [2], 51000.0 [3], 530000.0 [4]
F-AmidineKi330000.0 [1]
2-{[(2s)-1-Amino-5-{[(1z)-2-Fluoroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic AcidIC50400.0 [1], 1100.0 [2], 4600.0 [3], 32000.0 [4]
2-{[(2s)-1-Amino-5-{[(1z)-2-Fluoroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic AcidKi16000.0 [1]
2-{[(2s)-1-Amino-5-{[(1z)-2-Chloroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic AcidIC501100.0 [1], 2400.0 [2], 5300.0 [3], 22000.0 [4]
2-{[(2s)-1-Amino-5-{[(1z)-2-Chloroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic AcidKi13000.0 [1]
MinocyclineIC50620000.0 [1]
MinocyclineKi180000.0 [1], 540000.0 [2]
ChlortetracyclineIC50100000.0 [1]
ChlortetracyclineKi110000.0 [1], 540000.0 [2]
StreptomycinIC501800000.0 [1]
StreptomycinKi560000.0 [1]
DoxycyclineIC50860000.0 [1]
DoxycyclineKi630000.0 [1]
MethotrexateIC5010000000.0 [1]
TetracyclineIC50780000.0 [1]
AzathioprineIC508100000.0 [1]
ClindamycinIC505100000.0 [1]
AzithromycinIC5010000000.0 [1]
TrimethoprimIC507500000.0 [1]
SulfamethoxazoleIC5010000000.0 [1]
MesalamineIC5010000000.0 [1]
LeflunomideIC502400000.0 [1]
SulfapyridineIC5010000000.0 [1]
StreptonigrinIC502500.0 [1]
Cl-amidineIC505900.0 [1]
7-Amino-2-pyridin-2-ylquinoline-5,8-dioneIC50640.0 [1]
7-Bromo-6-methoxyquinoline-5,8-dioneIC503300.0 [1]
6-(7-Amino-5,8-dioxo-5,8-dihydroquinolin-2-yl)picolinic acidIC50240.0 [1]
7-Aminoquinoline-5,8-dioneIC501000.0 [1]
5,5-Dimethyl-3-(piperazin-1-ylmethyl)imidazolidine-2,4-dioneKi183000.0 [1]
[(3S,4R)-3-Amino-4-hydroxypiperidin-1-yl]-[7-methoxy-1-methyl-2-[1-(2,2,2-trifluoroethyl)indol-2-yl]benzimidazol-5-yl]methanoneIC5079.43 [1]
[(3R)-3-Aminopiperidin-1-yl]-[2-(1-ethylindol-2-yl)-7-methoxy-1-methylbenzimidazol-5-yl]methanoneIC50100.0 [1]
[(3R)-3-Aminopiperidin-1-yl]-[7-methoxy-1-methyl-2-[1-(2,2,2-trifluoroethyl)indol-2-yl]benzimidazol-5-yl]methanoneIC5050.12 [1]
[(3R)-3-Aminopiperidin-1-yl]-[2-[1-(cyclopropylmethyl)indol-2-yl]-7-methoxy-1-methylbenzimidazol-5-yl]methanoneIC5039.81 [1]
[(3R)-3-Aminopiperidin-1-yl]-[1-methyl-2-[1-(2,2,2-trifluoroethyl)indol-2-yl]benzimidazol-5-yl]methanoneIC50158.49 [1]
[(3R)-3-Aminopiperidin-1-yl]-[2-[1-(cyclopropylmethyl)indol-2-yl]-1-methylbenzimidazol-5-yl]methanoneIC50125.89 [1]
N-[(2S)-4-(4-Methylpiperazin-1-yl)-1-oxo-1-(propan-2-ylamino)butan-2-yl]furan-2-carboxamideKi488000.0 [1]
N-[(2S)-1-(Benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]furan-2-carboxamideKi2823000.0 [1]
N-[(2S)-4-(4-Methylpiperazin-1-yl)-1-oxo-1-(propan-2-ylamino)butan-2-yl]cyclohexanecarboxamideKi10000000.0 [1]
N-[(2S)-1-(Benzylamino)-4-imidazol-1-yl-1-oxobutan-2-yl]furan-2-carboxamideKi10000000.0 [1]
N-[(2S)-4-(4-Methylpiperazin-1-yl)-1-oxo-1-(propan-2-ylamino)butan-2-yl]morpholine-4-carboxamideKi10000000.0 [1]
N-[(2S)-1-(Benzylamino)-4-imidazol-1-yl-1-oxobutan-2-yl]-1-methylpyrrole-2-carboxamideKi180000.0 [1]
N-[(2S)-4-[4-(Cyanomethyl)imidazol-1-yl]-1-oxo-1-(propan-2-ylamino)butan-2-yl]furan-2-carboxamideKi591000.0 [1]
5,5-Dimethyl-3-[2-(2H-tetrazol-5-yl)ethyl]imidazolidine-2,4-dioneKi47000.0 [1]
N-[(2S)-1-(Benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]-1-methylpyrrole-2-carboxamideKi64000.0 [1]
N-[(2S)-4-Imidazol-1-yl-1-oxo-1-(propan-2-ylamino)butan-2-yl]furan-2-carboxamideKi88000.0 [1]
N'-[3-(1-Benzylindol-3-yl)propyl]-2-chloroethanimidamideIC5029000.0 [1]
2-Chloro-N'-[3-[1-(cyclopentylmethyl)indazol-3-yl]propyl]ethanimidamideIC5016000.0 [1]
2-Chloro-N'-[3-[1-(cyclopentylmethyl)indol-3-yl]propyl]ethanimidamideIC5021000.0 [1]
2-Chloro-N'-[3-(1-methylindol-3-yl)propyl]ethanimidamideIC50190000.0 [1]
2-Chloro-N'-[3-(1-ethylindol-3-yl)propyl]ethanimidamideIC5036000.0 [1]
5,5-Dimethyl-3-(2-morpholin-4-ylethyl)imidazolidine-2,4-dioneKi1430000.0 [1]
2-Fluoroacetimidamide hydrochlorideIC5010000000.0 [1]
5,5-Dimethyl-3-(2-pyrrolidin-1-ylethyl)imidazolidine-2,4-dioneKi4643000.0 [1]
3-(2-Imidazol-1-ylethyl)-5,5-dimethylimidazolidine-2,4-dioneKi632000.0 [1]
7-Amino-6-bromoquinoline-5,8-dioneIC50560.0 [1]
(2S)-5-[(1-Amino-2-fluoroethylidene)amino]-2-(benzenesulfonamido)pentanamideIC50500000.0 [1]
N-[(2S)-1-Amino-5-[(1-amino-2-fluoroethylidene)amino]-1-oxopentan-2-yl]-1H-imidazole-5-carboxamideIC50230000.0 [1]
N-[(2S)-1-Amino-5-[(1-amino-2-fluoroethylidene)amino]-1-oxopentan-2-yl]-1H-pyrrole-3-carboxamideIC5019000.0 [1]
N-[(2S)-1-Amino-5-[(1-amino-2-fluoroethylidene)amino]-1-oxopentan-2-yl]-2-hydroxy-5-nitrobenzamideIC5012000.0 [1]
2-Fluoro-N'-propylethanimidamideIC501000000.0 [1]
N'-Benzyl-2-fluoroethanimidamideIC501000000.0 [1]
2-Fluoro-N'-phenylethanimidamideIC50500000.0 [1]
N-[(2S)-1-Amino-3-[3-[(1-amino-2-fluoroethylidene)amino]phenyl]-1-oxopropan-2-yl]benzamideIC50310000.0 [1]
N-[(1S)-2-Amino-1-[3-[(1-amino-2-fluoroethylidene)amino]phenyl]-2-oxoethyl]benzamideIC502100000.0 [1]
N-[(2S)-1-Amino-3-[4-[(1-amino-2-fluoroethylidene)amino]phenyl]-1-oxopropan-2-yl]benzamideIC50310000.0 [1]
N-[(2S)-1-Amino-3-[4-[[(1-amino-2-fluoroethylidene)amino]methyl]phenyl]-1-oxopropan-2-yl]benzamideIC501000000.0 [1]
N-[4-[(1-Amino-2-fluoroethylidene)amino]butyl]benzamideIC501000000.0 [1]
N'-[4-(Benzenesulfonamido)butyl]-2-fluoroethanimidamideIC501000000.0 [1]
Items per page: 1 - 10 of 72
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein-arginine deiminase type-4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Protein-arginine deiminase type-4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-4-inhibitors-ic50-ki.
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