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Protein-arginine deiminase type-4 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Cl-amidine (TFA)IC503400.0 [1], 4000.0 [2], 9000.0 [3], 15000.0 [4]
Cl-amidine (TFA)Ki180000.0 [1]
F-AmidineIC5015000.0 [1], 21000.0 [2], 51000.0 [3], 530000.0 [4]
F-AmidineKi330000.0 [1]
2-{[(2s)-1-Amino-5-{[(1z)-2-Fluoroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic AcidIC50400.0 [1], 1100.0 [2], 4600.0 [3], 32000.0 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseProtein-arginine deiminase type-4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-4-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseProtein-arginine deiminase type-4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-4-inhibitors-ic50-ki.
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