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Protein kinase C (PKC) Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
StaurosporineIC506.0 [1]
Antibiotic K 252aIC5025.0 [1], 33.0 [2], 60.0 [3], 250.0 [4]
Arcyriaflavin aIC50310.0 [1], 550.0 [2], 44700.0 [3], 100000.0 [4]
6,7,12,13-Tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-oneIC502450.0 [1]
TamoxifenIC501000.0 [1], 20000.0 [2]
AlvocidibIC5010000.0 [1], 15000.0 [2]
RebeccamycinIC50100000.0 [1], 175000.0 [2]
5-[(2S)-2-Methylpiperazin-1-yl]sulfonylisoquinolineIC506000.0 [1]
5-[(2S)-2-Methylpiperazin-1-yl]sulfonylisoquinolineKi6000.0 [1]
1-(5-Isoquinolinesulfonyl)-2-methylpiperazine dihydrochlorideIC506000.0 [1]
1-(5-Isoquinolinesulfonyl)-2-methylpiperazine dihydrochlorideKi6000.0 [1]
(2S)-5-(Diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-3-hydroxy-2-[3-[2-(isoquinolin-5-ylsulfonylamino)ethylamino]propanoylamino]propanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoic acidIC50300.0 [1]
(2S)-5-(Diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-3-hydroxy-2-[3-[2-(isoquinolin-5-ylsulfonylamino)ethylamino]propanoylamino]propanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoic acidKi100.0 [1]
(2S)-5-(Diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-(isoquinolin-5-ylsulfonylamino)propanoyl]amino]propanoyl]amino]propanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoic acidIC507000.0 [1]
(2S)-5-(Diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-(isoquinolin-5-ylsulfonylamino)propanoyl]amino]propanoyl]amino]propanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoyl]amino]pentanoic acidKi8000.0 [1]
SuraminIC5029000.0 [1]
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazoleIC5075000.0 [1]
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamideKi31700.0 [1]
HarmineIC50250000.0 [1]
9H-Pyrido[3,4-B]indoleIC5025000.0 [1]
K252aIC50250.0 [1]
Methyl (15S,16S,18R)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8,10,12,20,22,24,26-nonaene-16-carboxylateIC50114.0 [1]
Bisindolylmaleimide IXIC5010.0 [1]
Bisindolylmaleimide IVIC50190.0 [1]
TaxifolinIC50100000.0 [1]
4'-N-BenzoylstaurosporineIC5050.0 [1]
(2S,3R,4R,6R,18S)-18-Hydroxy-3-methoxy-2-methyl-4-(methylamino)-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-16-oneIC504.1 [1]
(2R,3S,4S,6S,18R)-18-Hydroxy-3-methoxy-2-methyl-4-(methylamino)-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-16-oneIC5013.0 [1]
N-(2-(Methylamino)ethyl)-5-isoquinolinesulfonamideKi15000.0 [1]
CorilaginIC5020000.0 [1]
PentagalloylglucoseIC504000.0 [1]
MinaprineIC50100000.0 [1]
3-[(8S)-8-[(Dimethylamino)methyl]-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC5017.2 [1]
4,5-DianilinophthalimideIC5080000.0 [1]
N-(6-Chloro-9h-pyrido[3,4-b]indol-8-yl)-3-pyridinecarboxamideIC5025000.0 [1]
N-(2-Aminoethyl)isoquinoline-5-sulfonamideIC507000.0 [1]
Chebulagic acidIC5030000.0 [1]
beta-GlucogallinIC50100000.0 [1]
BalanolKi5.3 [1]
5,6-Bis[(4-fluorophenyl)amino]-1H-isoindole-1,3(2H)-dioneIC5032000.0 [1]
(46S)-7,8,9,12,13,14,25,26,27,30,31,32,35,36,37,46-Hexadecahydroxy-3,18,21,41,43-pentaoxanonacyclo[27.13.3.138,42.02,20.05,10.011,16.023,28.033,45.034,39]hexatetraconta-5,7,9,11,13,15,23,25,27,29(45),30,32,34(39),35,37-pentadecaene-4,17,22,40,44-pentoneIC504000.0 [1]
CastalaginIC508000.0 [1]
EdotecarinIC50200000.0 [1]
2-O-Methyl-PAF (C)IC5012000.0 [1]
Unii-NA856793UTIC5050000.0 [1]
4-Amino-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-7-Yl-CyclopentaneIC5033000.0 [1]
[(2R,3R,4R)-3,4,5-Trihydroxy-4-[(3,4,5-trihydroxybenzoyl)oxymethyl]oxolan-2-yl]methyl 3,4,5-trihydroxybenzoateIC50100000.0 [1]
(5R,6R,13S,21R)-5,13-Bis(3,4-dihydroxyphenyl)-4,12,14-trioxapentacyclo[11.7.1.02,11.03,8.015,20]henicosa-2(11),3(8),9,15,17,19-hexaene-6,9,17,19,21-pentolIC50100000.0 [1]
7-[cis-4-(4-Methylpiperazin-1-Yl)cyclohexyl]-5-(4-Phenoxyphenyl)-7h-Pyrrolo[2,3-D]pyrimidin-4-AmineIC5020000.0 [1]
1-(5-Isoquinolinesulfonyl)piperazineIC5012000.0 [1]
1-Tert-butyl-3-[6-(2,6-dichlorophenyl)-2-[4-(diethylamino)butylamino]pyrido[2,3-d]pyrimidin-7-yl]ureaIC5023000.0 [1]
A-770041IC5025000.0 [1]
9-Hydroxy-4-phenyl-6H-pyrrolo[3,4-C]carbazole-1,3-dioneIC503400.0 [1]
3,4,5-Tri-O-galloylquinic acidIC50100000.0 [1]
1,2,6-TrigalloylglucoseIC50100000.0 [1]
Bms-509744IC5024000.0 [1]
LetaxabanIC5060000.0 [1]
3,3'-Digalloylprocyanidin B2IC504000.0 [1]
Procyanidin C1IC5040000.0 [1]
Tpl2 Kinase InhibitorIC50400000.0 [1]
2-[4-(3-Phenylquinoxalin-2-yl)phenyl]propan-2-amineIC50250000.0 [1]
PDGF Receptor Tyrosine Kinase Inhibitor IIIIC5030000.0 [1]
4,5-Bis-(4-methoxyanilino)phthalimideIC50460000.0 [1]
1,3,4,5-Tetra-O-galloylquinic acidIC5064000.0 [1]
N-(3-Bromophenyl)-1H-imidazo[4,5-g]quinazolin-8-amineIC5050000.0 [1]
1,6-Bis-O-galloyl-beta-D-glucoseIC50100000.0 [1]
1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylureaIC5050000.0 [1]
10-Chlorobenzo[c]quinolizin-11-ium-6-olIC5038000.0 [1]
3-[(2R,3R,4R,5S,6R)-3,4-Dihydroxy-6-(hydroxymethyl)-5-methoxyoxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17,19,21-nonaene-12,14-dioneIC50142000.0 [1]
4-[(3-Chloro-4-fluorophenyl)amino]-6-[(1H-imidazol-4-ylmethyl)amino]quinoline-3-carbonitrileIC5010000.0 [1]
N'-(Pyrrolidino[2,1-B]isoindolin-4-ON-8-YL)-N-(pyridin-2-YL)ureaIC5020000.0 [1]
3,5-Di-O-galloylshikimic acidIC50100000.0 [1]
4-[3-Methyl-2-piperidin-4-yl-5-[3-(trifluoromethyl)phenyl]imidazol-4-yl]-N-[(1S)-1-phenylethyl]pyridin-2-amineIC501500.0 [1]
3-[(2R,3R,4R,5S,6R)-3,4-Dihydroxy-6-(hydroxymethyl)-5-methoxyoxan-2-yl]-13-methyl-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17,19,21-nonaene-12,14-dioneIC50100000.0 [1]
2-(2-Chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-chromen-4-oneIC50160000.0 [1]
(2R,3S,4S,6S)-4-Hydroxy-3-methoxy-2-methyl-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-16-oneIC503000.0 [1]
4-(3-Chloro-4-fluoro-phenylamino)-6-(2-morpholin-4-yl-ethylamino)-1,7-naphthyridine-3-carbonitrileIC5030000.0 [1]
4-[3-Methyl-2-piperidin-4-yl-5-[3-(trifluoromethyl)phenyl]imidazol-4-yl]-N-[(1S)-1-phenylethyl]pyrimidin-2-amineIC506000.0 [1]
14-Hydroxy-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4,6,8,10,15,17,19,21-nonaen-12-oneIC5022100.0 [1]
Unii-8FX9DP2Y1WIC5010000.0 [1]
4-(6,7-Dimethoxy-4-quinazolinyl)-N-(4-nitrophenyl)-1-piperazinecarboxamideIC5030000.0 [1]
n-Methyl-4,5-dianilinophthalimideIC50100000.0 [1]
5,21-Dichloro-3-[(2R,3R,4R,5S,6R)-3,4-dihydroxy-6-(hydroxymethyl)-5-methoxyoxan-2-yl]-13-methyl-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dioneIC50100000.0 [1]
N-Benzyl-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamideIC5030000.0 [1]
[(2R,3R,4S,5R,6R)-6-Hydroxy-3,4,5-tris[(3,4,5-trihydroxybenzoyl)oxy]oxan-2-yl]methyl 3,4,5-trihydroxybenzoateIC5082000.0 [1]
Eudistomin NIC5025000.0 [1]
13-(1,3-Dihydroxypropan-2-ylamino)-5,21-dihydroxy-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dioneIC50200000.0 [1]
PunicafolinIC504000.0 [1]
6-Acetyl-8-cyclopentyl-5-methyl-2-(4-piperazin-1-yl-phenylamino)-8H-pyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
Dichloroarcyriaflavin AIC5050000.0 [1]
6-Methoxy-9H-pyrido[3,4-b]indoleIC5025000.0 [1]
N-(1,3-Benzodioxol-5-ylmethyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carbothioamideIC5030000.0 [1]
(15R,16R,18S)-16-(Hydroxymethyl)-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8,10,12,20,22,24,26-nonaene-3,5-dioneIC501.7 [1]
5-[(4-Aminopiperidin-1-yl)methyl]-N-[1-[(3-fluorophenyl)methyl]indazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-4-amineIC502200.0 [1]
N-(4-Bromophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamideIC5030000.0 [1]
N-(4-Cyanophenyl)-4-(6,7-dimethoxyquinazolin-4-yl)piperazine-1-carboxamideIC5030000.0 [1]
4-(6,7-Dimethoxyquinazolin-4-yl)-N-(4-propan-2-ylphenyl)piperazine-1-carboxamideIC5030000.0 [1]
6,8-Dichloro-9h-pyrido[3,4-b]indoleIC5025000.0 [1]
3-[[5-Cyano-6-(cyclopentylamino)pyrimidin-4-yl]amino]-4-methyl-N-(1,2-oxazol-3-yl)benzamideIC5050000.0 [1]
5-Bromo-6-methoxy-beta-carbolineIC5015000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein kinase C (PKC) Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/protein-kinase-c-pkc-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Protein kinase C (PKC) Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-kinase-c-pkc-inhibitors-ic50-ki.
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