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Protein-tyrosine phosphatase 2C Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
6-Hydroxy-1-methyl-3-[1-[3-oxo-3-(4-phenylanilino)propyl]triazol-4-yl]-2-phenylindole-5-carboxylic acidIC505500.0 [1], 9000.0 [2], 10800.0 [3]
6-Hydroxy-1-methyl-3-[1-[3-oxo-3-(4-phenylanilino)propyl]triazol-4-yl]-2-phenylindole-5-carboxylic acidKi5200.0 [1]
1-(2-Methyl-4,5-disulfophenyl)-5-oxo-4,5-dihydro-1H-pyrazole-3-carboxylic acidIC508300.0 [1], 26000.0 [2], 56000.0 [3]
1-(2-Methyl-4,5-disulfophenyl)-5-oxo-4,5-dihydro-1H-pyrazole-3-carboxylic acidKi4600.0 [1]
8-Hydroxy-7-(6-sulfo-naphthalen-2-ylazo)-quinoline-5-sulfonic acidIC50318.0 [1], 1110.0 [2]
2-Hydroxy-3-[(2-nitrophenyl)diazenyl]-1H-indole-5-sulfonic acidIC504990.0 [1], 46800.0 [2], 47260.0 [3]
SodiumIC50300.0 [1], 320.0 [2]
Oleanolic acidIC5011620.0 [1], 120000.0 [2]
CryptotanshinoneIC5022500.0 [1], 45180.0 [2]
Cefsulodin sodium saltIC5016800.0 [1]
Cefsulodin sodium saltKi6600.0 [1]
4-[5-[4-(4-Fluorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC5031900.0 [1]
3-[[5-[(4-Fluorophenyl)methylsulfamoyl]-2-hydroxy-1H-indol-3-yl]diazenyl]benzoic acidIC501000.0 [1]
4-(2-(3-(4-Nitrophenyl)-5-oxo-1-phenyl-1H-pyrazol-4(5H)-ylidene)hydrazinyl)benzenesulfonic acidIC502100.0 [1]
4-(2-(3-(4-Nitrophenyl)-5-oxo-1-phenyl-1H-pyrazol-4(5H)-ylidene)hydrazinyl)benzenesulfonic acidKi700.0 [1]
3-[2-(2-Nitrophenyl)hydrazinyl]indol-2-oneIC5060000.0 [1], 66500.0 [2]
(3S,3Ar,5S,6aR)-N-(cyclohexylmethyl)-3-[5-[3-(pyrrolidin-1-ylmethyl)phenyl]tetrazol-1-yl]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-5-amineIC502470.0 [1], 2500.0 [2]
3-[(3-Nitrophenyl)diazenyl]-1H-indol-2-olIC5060000.0 [1], 100000.0 [2]
2-[4-[[2-(4-Iodoanilino)-2-oxoacetyl]amino]anilino]-2-oxo-1-phenylethanesulfonic acidIC501500.0 [1]
2-[4-[[2-(4-Iodoanilino)-2-oxoacetyl]amino]anilino]-2-oxo-1-phenylethanesulfonic acidKi510.0 [1]
(3Z)-3-[2-(2-Nitrophenyl)hydrazin-1-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonamideIC504990.0 [1], 11900.0 [2]
(3Z)-3-[2-(3-Carboxyphenyl)hydrazin-1-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-carboxylic acidIC5015800.0 [1], 16070.0 [2]
3-[[5-[(4-Chlorophenyl)methylcarbamoyl]-2-hydroxy-1H-indol-3-yl]diazenyl]benzoic acidIC5022300.0 [1], 100000.0 [2]
3-{2-[(3Z)-2-Oxo-5-(propan-2-ylsulfamoyl)-2,3-dihydro-1H-indol-3-ylidene]hydrazin-1-yl}benzoic acidIC504500.0 [1], 7580.0 [2]
N-[(4-Chlorophenyl)methyl]-2-hydroxy-3-[(2-nitrophenyl)diazenyl]-1H-indole-5-sulfonamideIC504400.0 [1], 10120.0 [2]
(3Z)-3-[2-(2-Carboxyphenyl)hydrazin-1-ylidene]-2-oxo-2,3-dihydro-1H-indole-5-carboxylic acidIC50800.0 [1], 3550.0 [2]
5-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}-1-(cyclopropylcarbonyl)indolineIC508500.0 [1]
4-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC50700.0 [1], 37300.0 [2]
4-[5-[4-(5-Chloro-2-methylphenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC501500.0 [1]
US8623906, Jhe-02-069IC508200.0 [1]
N-(3-Chlorophenyl)-5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carboxamideIC508300.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(4-propan-2-ylphenyl)-2,3-dihydroindole-1-carboxamideIC504100.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(3,4-dichlorophenyl)-2,3-dihydroindole-1-carboxamideIC505700.0 [1]
4-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC502500.0 [1]
N-(2-Chlorophenyl)-5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carboxamideIC503200.0 [1]
5-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-5-oxopentanoic acidIC502800.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-(4-methoxyphenyl)methanoneIC506300.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-cyclopentylmethanoneIC506900.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]acetic acidIC504600.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-methylpentanoic acidIC5015500.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-(3,5-dichlorophenyl)methanoneIC508200.0 [1]
N-(4-Chlorophenyl)-5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carboxamideIC5019100.0 [1]
(3-Chlorophenyl)-[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]methanoneIC505700.0 [1]
1-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-3-methylbutan-1-oneIC5020700.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(3-methoxyphenyl)-2,3-dihydroindole-1-carboxamideIC509900.0 [1]
2-(4-Chlorophenyl)-1-[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]ethanoneIC508000.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-(2,4-dichlorophenyl)methanoneIC507600.0 [1]
4-[5-[4-(3,5-Dichlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC504500.0 [1]
4-[5-[4-[3,5-Bis(trifluoromethyl)phenyl]piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC509100.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(4-fluorophenyl)-2,3-dihydroindole-1-carboxamideIC5012600.0 [1]
Ethyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-4-methylpentanoateIC506000.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-(3-methoxyphenyl)methanoneIC508100.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-phenylmethanoneIC508400.0 [1]
[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-(3,4-dichlorophenyl)methanoneIC507100.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-methylbutanoic acidIC504400.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(3-fluorophenyl)-2,3-dihydroindole-1-carboxamideIC508100.0 [1]
Ethyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]propanoateIC505100.0 [1]
2-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-2-oxoacetic acidIC504800.0 [1]
1-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]butan-1-oneIC507800.0 [1]
3-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]propanoic acidIC504800.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-4-methylpentanoic acidIC504500.0 [1]
4-[5-[4-(3-Methoxyphenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC504700.0 [1]
Ethyl 3-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]propanoateIC509300.0 [1]
Methyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-methylpentanoateIC5012700.0 [1]
Ethyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-methylbutanoateIC507700.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-(2-fluorophenyl)-2,3-dihydroindole-1-carboxamideIC5012200.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-phenyl-2,3-dihydroindole-1-carboxamideIC5011700.0 [1]
5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-N-[2-(trifluoromethyl)phenyl]-2,3-dihydroindole-1-carboxamideIC509000.0 [1]
(4-Chlorophenyl)-[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]methanoneIC5010400.0 [1]
3-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]benzoic acidIC503000.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]benzoic acidIC508300.0 [1]
Methyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]benzoateIC5014300.0 [1]
1-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-2-methoxyethanoneIC509600.0 [1]
6-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]cyclohex-3-ene-1-carboxylic acidIC5020300.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-phenylpropanoic acidIC505400.0 [1]
4-[5-[4-(3-Chloro-4-methylphenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC5016600.0 [1]
1-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-2-phenylethanoneIC5022800.0 [1]
1-[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]-2,2,2-trifluoroethanoneIC5047000.0 [1]
4-[5-[4-(2-Fluorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC5034600.0 [1]
Ethyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]acetateIC5060300.0 [1]
US8623906, XW2-038AIC5014800.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]pentanedioic acidIC5037600.0 [1]
4-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC50143600.0 [1]
Ethyl 2-[[5-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]-3-phenylpropanoateIC506900.0 [1]
4-Oxo-4-[5-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]butanoic acidIC5011300.0 [1]
4-[5-[4-(4-Methoxyphenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC509000.0 [1]
4-[5-[4-(3,4-Dichlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC504600.0 [1]
4-[5-[4-(3-Fluorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]-4-oxobutanoic acidIC5013200.0 [1]
2-[[5-[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindole-1-carbonyl]amino]propanoic acidIC506400.0 [1]
1-[5-[4-(3-Methylphenyl)piperazin-1-yl]sulfonyl-2,3-dihydroindol-1-yl]propan-1-oneIC503400.0 [1]
EstradiolIC50300000.0 [1]
EnoxoloneIC509600.0 [1]
EstramustineIC50300000.0 [1]
Tanshinone IIAIC502590.0 [1]
Tanshinone IIC502570.0 [1]
Estramustine phosphateIC5017100.0 [1]
CelastrolIC503300.0 [1]
Maslinic acidIC5040000.0 [1]
Polyestradiol phosphateIC5019900.0 [1]
Pyrogallol RedIC502440.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein-tyrosine phosphatase 2C Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/protein-tyrosine-phosphatase-2c-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Protein-tyrosine phosphatase 2C Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-tyrosine-phosphatase-2c-inhibitors-ic50-ki.
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