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Proteinase-activated receptor 2 Inhibitors (IC50, Ki)
Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
 | N-[(2S)-3-Cyclohexyl-1-[[(2S,3S)-3-methyl-1-oxo-1-(4-phenylpiperidin-1-yl)pentan-2-yl]amino]-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide | IC50 | 2200.0 [1] |
 | N-[(2S)-3-Cyclohexyl-1-[[(2S,3S)-3-methyl-1-oxo-1-spiro[indene-1,4'-piperidine]-1'-ylpentan-2-yl]amino]-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide | IC50 | 1000.0 [1], 1584.89 [2], 3600.0 [3], 9600.0 [4] |
 | N-[(2S)-3-Cyclohexyl-1-[[(2S,3S)-1-[(2-methoxyphenyl)methylamino]-3-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide | IC50 | 400.0 [1], 500.0 [2], 1700.0 [3], 1900.0 [4] |
 | Tert-butyl 4-[8-tert-butyl-6-(4-fluorophenyl)imidazo[1,2-b]pyridazine-2-carbonyl]-3,3-dimethylpiperazine-1-carboxylate | IC50 | 4.2 [1], 4.8 [2], 50000.0 [3] |
 | Tert-butyl 4-[6-(4-fluorophenyl)-8-propan-2-ylimidazo[1,2-b]pyridazine-2-carbonyl]-3,3-dimethylpiperazine-1-carboxylate | IC50 | 2.0 [1], 5.0 [2], 51000.0 [3], 97000.0 [4] |
References
This online resource may be cited as follows
MLA | "Quest Database™ Proteinase-activated receptor 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2026, https://www.aatbio.com/data-sets/proteinase-activated-receptor-2-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, May 9). Quest Database™ Proteinase-activated receptor 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/proteinase-activated-receptor-2-inhibitors-ic50-ki. | |
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