Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 1-[(trans-4-Aminocyclohexyl)methyl]-N-Butyl-3-(4-Fluorophenyl)-1h-Pyrazolo[3,4-D]pyrimidin-6-Amine | IC50 | 2.9 [1], 141.0 [2] | |
| 1-[(trans-4-Aminocyclohexyl)methyl]-N-Butyl-3-(4-Fluorophenyl)-1h-Pyrazolo[3,4-D]pyrimidin-6-Amine | Ki | 4.3 [1] | |
| 2-(2-Hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | IC50 | 11000.0 [1], 11300.0 [2] | |
| 4-[2-(Butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 0.46 [1], 0.74 [2], 2.7 [3] | |
| 4-[5-[4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl]-2-[[(2S)-pentan-2-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | IC50 | 0.6 [1], 2.4 [2], 13.8 [3] | |
MLA | "Quest Database™ Proto-oncogene tyrosine-protein kinase MER Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 Feb. 2026, https://www.aatbio.com/data-sets/proto-oncogene-tyrosine-protein-kinase-mer-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, February 9). Quest Database™ Proto-oncogene tyrosine-protein kinase MER Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/proto-oncogene-tyrosine-protein-kinase-mer-inhibitors-ic50-ki. | |
| BibTeX | EndNote | RefMan |