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Purinergic receptor P2Y12 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
Ethyl 6-{4-[(Benzylsulfonyl)carbamoyl]piperidin-1-Yl}-5-Cyano-2-Methylpyridine-3-CarboxylateIC509.0 [1], 25.0 [2], 3200.0 [3]
1-(5-Butanoyl-3-cyano-6-methylsulfanylpyridin-2-yl)-N-(1-phenylcyclopropyl)sulfonylpiperidine-4-carboxamideIC501.0 [1], 19.0 [2], 640.0 [3]
Ethyl 6-[3-({[(5-chloro-2-thienyl)sulfonyl]amino}carbonyl)azetidin-1-yl]-5-cyano-2-methylnicotinateIC5068.0 [1], 22000.0 [2]
TicagrelorIC505.01 [1], 320.0 [2], 500.0 [3]
TicagrelorKi2.0 [1], 14.0 [2]
(4S)-4-[[4-[4-(Methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidIC501800.0 [1], 50000.0 [2]
(4S)-4-[[4-[4-(Methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidKi15.0 [1], 510.0 [2]
Ethyl 6-[4-({[(5-chloro-2-thienyl)sulfonyl]amino}carbonyl)piperazin-1-yl]-5-cyano-2-methylnicotinateIC5019.0 [1], 34.0 [2], 40.0 [3], 42.0 [4], 70.0 [5]
SodiumKi2100.0 [1], 2390.0 [2], 2450.0 [3], 17100.0 [4]
CangrelorIC500.4 [1], 2.0 [2], 18.3 [3]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidIC50770.0 [1]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidKi7.0 [1], 15.0 [2]
Ethyl 6-[4-(anilinocarbonyl)piperazin-1-yl]-5-cyanonicotinateIC50920.0 [1], 2600.0 [2]
Ethyl 5-chloro-6-(4-{[(4-methylphenyl)amino]carbonyl}piperazin-1-yl)nicotinateIC50600.0 [1], 1100.0 [2]
Ethyl 5-chloro-6-(4-{[(2-methylphenyl)amino]carbonyl}piperazin-1-yl)nicotinateIC501400.0 [1], 2600.0 [2]
Ethyl 5-cyano-6-[4-(phenylcarbamoyl)piperazin-1-yl]-2-(trifluoromethyl)pyridine-3-carboxylateIC50320.0 [1], 330.0 [2], 680.0 [3]
Ethyl 5-cyano-6-(4-{[(4-fluorobenzyl)amino]carbonyl}piperazin-1-yl)-2-(trifluoro-methyl)nicotinateIC50110.0 [1], 470.0 [2]
Ethyl 6-[4-(anilinocarbonyl)piperazin-1-yl]-5-chloronicotinateIC50880.0 [1], 890.0 [2], 1700.0 [3]
2-Methyl-5-cyano-6-[4-[(5-chloro-2-thienylsulfonyl)carbamoyl]piperidino]nicotinic acid ethyl esterIC5039.0 [1], 80.0 [2], 22000.0 [3]
ElinogrelIC5010.0 [1], 10000.0 [2]
ElinogrelKi23.0 [1]
Acid Blue 25IC503120.0 [1]
Acid Blue 25Ki9830.0 [1]
CID 16681707IC5029.0 [1], 130.0 [2]
CID 16681707Ki86.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(4-hydroxypiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC509800.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(4-hydroxypiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi42.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC508100.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi114.0 [1], 117.0 [2]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(3-hydroxypropoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC509000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(3-hydroxypropoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi68.0 [1]
(S)-5-Oxo-4-(6-phenylpicolinamido)-5-(4-m-tolylpiperazin-1-yl)pentanoic acidIC50100000.0 [1]
(S)-5-Oxo-4-(6-phenylpicolinamido)-5-(4-m-tolylpiperazin-1-yl)pentanoic acidKi5700.0 [1]
(S)-5-(4-(Heptyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidIC5056000.0 [1]
(S)-5-(4-(Heptyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidKi7.0 [1]
(S)-5-(4-(Ethoxycarbonyl)piperazin-1-yl)-4-(4-methoxy-6-phenylpicolinamido)-5-oxopentanoic acidIC5039000.0 [1]
(S)-5-(4-(Ethoxycarbonyl)piperazin-1-yl)-4-(4-methoxy-6-phenylpicolinamido)-5-oxopentanoic acidKi96.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC505800.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi92.0 [1], 140.0 [2]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC507600.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi157.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-oxo-5-(4-(pentyloxycarbonyl)piperazin-1-yl)pentanoic acidIC5028400.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-oxo-5-(4-(pentyloxycarbonyl)piperazin-1-yl)pentanoic acidKi49.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-5-oxo-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidIC501100.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-5-oxo-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidKi12.0 [1]
(S)-5-(4-(Octyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidIC50100000.0 [1]
(S)-5-(4-(Octyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidKi14.0 [1]
(4S)-4-[[4-(2-Hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidIC5011500.0 [1]
(4S)-4-[[4-(2-Hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidKi31.0 [1], 32.0 [2]
(S)-5-Oxo-5-(4-(pentyloxycarbonyl)piperazin-1-yl)-4-(6-phenylpicolinamido)pentanoic acidIC5015000.0 [1]
(S)-5-Oxo-5-(4-(pentyloxycarbonyl)piperazin-1-yl)-4-(6-phenylpicolinamido)pentanoic acidKi11.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidIC501900.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidKi68.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC507800.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-4-[[4-(2-hydroxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi20.0 [1], 21.0 [2]
(S)-4-(4,6-Diphenylpicolinamido)-5-oxo-5-(4-m-tolylpiperazin-1-yl)pentanoic acidIC50100000.0 [1]
(S)-4-(4,6-Diphenylpicolinamido)-5-oxo-5-(4-m-tolylpiperazin-1-yl)pentanoic acidKi5.7 [1], 150.0 [2]
(4S)-4-[[4-(2-Aminoethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidIC507500.0 [1]
(4S)-4-[[4-(2-Aminoethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidKi328.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(methylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC5045000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(methylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi35.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC5014000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethylamino)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi99.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-(4-(ethoxycarbonyl)piperazin-1-yl)-5-oxopentanoic acidIC5033900.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-(4-(ethoxycarbonyl)piperazin-1-yl)-5-oxopentanoic acidKi39.0 [1], 60.0 [2]
(4S)-4-[[4-(4-Aminopiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidIC502800.0 [1]
(4S)-4-[[4-(4-Aminopiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidKi10.0 [1], 27.0 [2]
(S)-5-Oxo-4-(6-phenylpicolinamido)-5-(4-(propoxycarbonyl)piperazin-1-yl)pentanoic acidIC5062000.0 [1]
(S)-5-Oxo-4-(6-phenylpicolinamido)-5-(4-(propoxycarbonyl)piperazin-1-yl)pentanoic acidKi27.0 [1]
(S)-5-(4-(Hexyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidIC5019000.0 [1]
(S)-5-(4-(Hexyloxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidKi43.0 [1]
(4S)-4-[[4-(4-Hydroxypiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidIC502400.0 [1]
(4S)-4-[[4-(4-Hydroxypiperidin-1-yl)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidKi11.0 [1]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-(4-hexoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidIC501600.0 [1]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-(4-hexoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidKi18.0 [1]
(S)-5-(4-(Methoxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidIC50100000.0 [1]
(S)-5-(4-(Methoxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidKi2440.0 [1]
(S)-5-(4-(Butoxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidIC5028000.0 [1]
(S)-5-(4-(Butoxycarbonyl)piperazin-1-yl)-5-oxo-4-(6-phenylpicolinamido)pentanoic acidKi29.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC504400.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-4-[[4-(2-methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi18.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(4-pyrrolidin-1-ylpiperidin-1-yl)pyridine-2-carbonyl]amino]pentanoic acidIC502000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(4-pyrrolidin-1-ylpiperidin-1-yl)pyridine-2-carbonyl]amino]pentanoic acidKi34.0 [1]
(4S)-4-[[4-(2-Methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidIC504300.0 [1]
(4S)-4-[[4-(2-Methoxyethoxy)-6-phenylpyridine-2-carbonyl]amino]-5-oxo-5-(4-pentoxycarbonylpiperazin-1-yl)pentanoic acidKi9.9 [1], 10.0 [2]
(4S)-5-Oxo-5-(4-pentoxycarbonylpiperazin-1-yl)-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidIC50550.0 [1]
(4S)-5-Oxo-5-(4-pentoxycarbonylpiperazin-1-yl)-4-[(6-phenyl-4-piperidin-4-yloxypyridine-2-carbonyl)amino]pentanoic acidKi3.5 [1], 3.8 [2]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-[4-(methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC509900.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-4-[[4-[4-(methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi18.0 [1]
(4S)-5-(4-Hexoxycarbonylpiperazin-1-yl)-4-[[4-[4-(methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC507600.0 [1]
(4S)-5-(4-Hexoxycarbonylpiperazin-1-yl)-4-[[4-[4-(methoxymethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidKi33.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(piperidin-4-ylmethoxy)pyridine-2-carbonyl]amino]pentanoic acidIC504000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(piperidin-4-ylmethoxy)pyridine-2-carbonyl]amino]pentanoic acidKi76.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(propylamino)pyridine-2-carbonyl]amino]pentanoic acidIC5028000.0 [1]
(4S)-5-(4-Ethoxycarbonylpiperazin-1-yl)-5-oxo-4-[[6-phenyl-4-(propylamino)pyridine-2-carbonyl]amino]pentanoic acidKi64.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-(4-(butoxycarbonyl)piperazin-1-yl)-5-oxopentanoic acidIC5026900.0 [1]
(S)-4-(4-Butoxy-6-phenylpicolinamido)-5-(4-(butoxycarbonyl)piperazin-1-yl)-5-oxopentanoic acidKi35.0 [1], 36.0 [2]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidIC503300.0 [1]
(4S)-4-[[4-[4-(Aminomethyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acidKi14.0 [1]
(4S)-5-(4-Butoxycarbonylpiperazin-1-yl)-4-[[4-[4-(ethylcarbamoyl)piperidin-1-yl]-6-phenylpyridine-2-carbonyl]amino]-5-oxopentanoic acidIC50490.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Purinergic receptor P2Y12 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/purinergic-receptor-p2y12-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Purinergic receptor P2Y12 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/purinergic-receptor-p2y12-inhibitors-ic50-ki.
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