Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Ethyl 6-{4-[(Benzylsulfonyl)carbamoyl]piperidin-1-Yl}-5-Cyano-2-Methylpyridine-3-Carboxylate | IC50 | 9.0 [1], 25.0 [2], 3200.0 [3] | |
| 1-(5-Butanoyl-3-cyano-6-methylsulfanylpyridin-2-yl)-N-(1-phenylcyclopropyl)sulfonylpiperidine-4-carboxamide | IC50 | 1.0 [1], 19.0 [2], 640.0 [3] | |
| Ethyl 6-[3-({[(5-chloro-2-thienyl)sulfonyl]amino}carbonyl)azetidin-1-yl]-5-cyano-2-methylnicotinate | IC50 | 68.0 [1], 22000.0 [2] | |
| Ticagrelor | IC50 | 5.01 [1], 320.0 [2], 500.0 [3] | |
| Ticagrelor | Ki | 2.0 [1], 14.0 [2] | |
MLA | "Quest Database™ Purinergic receptor P2Y12 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 Jan. 2026, https://www.aatbio.com/data-sets/purinergic-receptor-p2y12-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, January 10). Quest Database™ Purinergic receptor P2Y12 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/purinergic-receptor-p2y12-inhibitors-ic50-ki. | |
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