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Pyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
(3S)-3-Amino-4-[4-[[2-(2,4-dihydroxyphenyl)sulfonyl-1,3-dihydroisoindol-5-yl]amino]piperidin-1-yl]-4-oxobutanamideIC501710.0 [1], 45800.0 [2]
Dichloroacetic acidIC505560000.0 [1]
RadicicolIC50230000.0 [1]
Dimorpholinethiuram disulfideKi2851.0 [1]
CID 86280454IC5040.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabasePyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.14 Dec2025https://www.aatbio.com/data-sets/pyruvate-dehydrogenase-kinase-isoform-3-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 14). Quest DatabasePyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pyruvate-dehydrogenase-kinase-isoform-3-inhibitors-ic50-ki.
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