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Pyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ShikoninIC508820.0 [1]
5-(2,5-Dimethyl-pyrrol-1-yl)-2-hydroxy-benzoic acidIC507000.0 [1], 12500.0 [2], 100000.0 [3]
ScutellareinIC5012500.0 [1], 100000.0 [2]
3-[2-(1H-Indol-3-yl)ethyl]-6-nitro-1H-indoleIC5054600.0 [1], 95900.0 [2]
[1,4-Dioxo-3-(piperidine-1-carbothioylsulfanylmethyl)naphthalen-2-yl]methyl piperidine-1-carbodithioateIC50880.0 [1], 5070.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabasePyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.18 Dec2025https://www.aatbio.com/data-sets/pyruvate-kinase-isozymes-m1-m2-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 18). Quest DatabasePyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pyruvate-kinase-isozymes-m1-m2-inhibitors-ic50-ki.
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