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Receptor-interacting serine/threonine-protein kinase 3 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
CID 67469084IC5016.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
(Arylindolyl)maleimide deriv. 27IC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-naphthalen-1-yl-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC50880.0 [1]
2-(6-Methoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC501200.0 [1]
2-(6-Ethoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC501700.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC502500.0 [1]
2-(1,3-Benzodioxol-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC507600.0 [1]
[3-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanoneIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-3-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-phenylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC505500.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-a]pyridineIC5010000.0 [1]
2-(2,3-Dihydro-1,4-benzodioxin-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(4-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(3-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC50450.0 [1]
6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-2-ylphenyl)imidazo[1,2-b]pyridazineIC50270.0 [1]
6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-3-ylphenyl)imidazo[1,2-b]pyridazineIC50300.0 [1]
2-(2,3-Dihydro-1,4-benzodioxin-6-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(5-phenylthiophen-2-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
[4-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanoneIC5010000.0 [1]
6-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]-1,3-benzothiazoleIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1H-indol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acidIC5010000.0 [1]
4-Hydroxy-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8,10,12,22,24,26-nonaene-3,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-1-hydroxy-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3,4-bis(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
1-Hydroxy-3-(1-methylindol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acidIC5010000.0 [1]
2-(3-Methoxyphenyl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Receptor-interacting serine/threonine-protein kinase 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/receptor-interacting-serine-threonine-protein-kinase-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Receptor-interacting serine/threonine-protein kinase 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/receptor-interacting-serine-threonine-protein-kinase-3-inhibitors-ic50-ki.
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