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Regulator of G-protein signaling 4 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
4-(4-Fluorobenzyl)-2-p-tolyl-1,2,4-thiadiazolidine-3,5-dioneIC5030.0 [1], 30.1 [2]
Unii-9egb3J3KI5IC50100000.0 [1]
1-Benzyl-3-p-tolyl-1H-pyrrole-2,5-dioneIC5093000.0 [1], 93300.0 [2]
4-Butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dioneIC5014.4 [1]
RGS4 inhibitor 13IC5054.3 [1]
4-Benzyl-2-phenyl-1,2,4-thiadiazolidine-3,5-dioneIC5023.5 [1]
4-Benzyl-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5023.9 [1]
4-Benzyl-2-(4-methyl-benzyl)-[1,2,4]thiadiazolidine-3,5-dioneIC507.2 [1]
2-Ethyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5022.3 [1]
2-Butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5023.5 [1]
2,4-Dibutyl-1,2,4-thiadiazolidine-3,5-dioneIC5029.8 [1]
4-[(4-Methoxyphenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC50176.0 [1]
4-[(4-Fluorophenyl)methyl]-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC50121.0 [1]
2-(3-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5052.3 [1]
2-(4-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5013.5 [1]
2-Butyl-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5015.6 [1]
4-Benzyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5014.4 [1]
4-Benzyl-2-(4-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5028.7 [1]
4-Benzyl-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dioneIC5057.4 [1]
4-[(4-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC505.4 [1]
4-[(3-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5017.4 [1]
4-[(3,4-Dichlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5034.2 [1]
4-Butyl-2-tert-butyl-1,2,4-thiadiazolidine-3,5-dioneIC5053.6 [1]
2-Ethyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5026.3 [1]
2-Tert-butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5029.1 [1]
4-[(4-Fluorophenyl)methyl]-2-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5012.9 [1]
2-(4-Methylphenyl)-4-[(3-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5014.5 [1]
2-(4-Methylphenyl)-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5014.0 [1]
2-Butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5038.6 [1]
2-(3,4-Dichlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5035.7 [1]
4-Benzyl-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5038.2 [1]
2-(4-Methylphenyl)-4-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC508.6 [1]
4-[(4-Fluorophenyl)methyl]-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5010.9 [1]
2-Tert-butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5027.8 [1]
4-[(4-Fluorophenyl)methyl]-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dioneIC5079.3 [1]
4-Benzyl-2-(3,4-dichlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5088.9 [1]
4-Methyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5018.9 [1]
4-[(4-Fluorophenyl)methyl]-2-phenyl-1,2,4-thiadiazolidine-3,5-dioneIC5016.3 [1]
4-Butyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5019.7 [1]
4-Benzyl-2-(3-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5032.5 [1]
2-Ethyl-4-(4-fluorobenzyl)-1,2,4-thiadiazolidine-3,5-dioneIC5022.3 [1]
1-Benzyl-3-bromo-1H-pyrrole-2,5-dioneIC5032000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Regulator of G-protein signaling 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/regulator-of-g-protein-signaling-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Regulator of G-protein signaling 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/regulator-of-g-protein-signaling-4-inhibitors-ic50-ki.
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