logo
AAT Bioquest

Regulator of G-protein signaling 8 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
4-(4-Fluorobenzyl)-2-p-tolyl-1,2,4-thiadiazolidine-3,5-dioneIC5011000.0 [1]
Unii-9egb3J3KI5IC50100000.0 [1]
1-Benzyl-3-p-tolyl-1H-pyrrole-2,5-dioneIC500.0 [1], 100000.0 [2]
4-Butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dioneIC5083500.0 [1]
RGS4 inhibitor 13IC5036100.0 [1]
4-Benzyl-2-phenyl-1,2,4-thiadiazolidine-3,5-dioneIC505600.0 [1]
4-Benzyl-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5012300.0 [1]
4-Benzyl-2-(4-methyl-benzyl)-[1,2,4]thiadiazolidine-3,5-dioneIC5020400.0 [1]
2-Ethyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5037000.0 [1]
2-Butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5028400.0 [1]
2,4-Dibutyl-1,2,4-thiadiazolidine-3,5-dioneIC50122000.0 [1]
4-[(4-Methoxyphenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC50312000.0 [1]
4-[(4-Fluorophenyl)methyl]-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC507100.0 [1]
2-(3-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5012800.0 [1]
2-(4-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC507600.0 [1]
2-Butyl-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5031600.0 [1]
4-Benzyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC507500.0 [1]
4-Benzyl-2-(4-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC505200.0 [1]
4-Benzyl-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dioneIC5016400.0 [1]
4-[(4-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5011800.0 [1]
4-[(3-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5017500.0 [1]
4-[(3,4-Dichlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5015700.0 [1]
4-Butyl-2-tert-butyl-1,2,4-thiadiazolidine-3,5-dioneIC50119000.0 [1]
2-Ethyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5070600.0 [1]
2-Tert-butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC50194000.0 [1]
4-[(4-Fluorophenyl)methyl]-2-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5039800.0 [1]
2-(4-Methylphenyl)-4-[(3-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC509900.0 [1]
2-(4-Methylphenyl)-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC507700.0 [1]
2-Butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dioneIC5098000.0 [1]
2-(3,4-Dichlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5017200.0 [1]
4-Benzyl-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5021300.0 [1]
2-(4-Methylphenyl)-4-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dioneIC5011600.0 [1]
4-[(4-Fluorophenyl)methyl]-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5011400.0 [1]
2-Tert-butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dioneIC5056000.0 [1]
4-[(4-Fluorophenyl)methyl]-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dioneIC5016200.0 [1]
4-Benzyl-2-(3,4-dichlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5013200.0 [1]
4-Methyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC508400.0 [1]
4-[(4-Fluorophenyl)methyl]-2-phenyl-1,2,4-thiadiazolidine-3,5-dioneIC506200.0 [1]
4-Butyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dioneIC509500.0 [1]
4-Benzyl-2-(3-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dioneIC5010900.0 [1]
2-Ethyl-4-(4-fluorobenzyl)-1,2,4-thiadiazolidine-3,5-dioneIC5018700.0 [1]
1-Benzyl-3-bromo-1H-pyrrole-2,5-dioneIC50100000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Regulator of G-protein signaling 8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/regulator-of-g-protein-signaling-8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Regulator of G-protein signaling 8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/regulator-of-g-protein-signaling-8-inhibitors-ic50-ki.
BibTeXEndNoteRefMan