Name: Renin Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Renin Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Aliskiren	IC50	0.6 ^[1]
	Pepstatin	IC50	6000.0 ^[1]
	Pepstatin	Ki	100.0 ^[1], 13000.0 ^[2]
	(2S)-1-[(2S)-2-[[(2S)-2-Amino-2-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]-N-[(2S)-1-[[(2S)-1-[[1-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-6-methyl-1-oxoheptan-4-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide	IC50	3.0 ^[1], 13.0 ^[2], 31.0 ^[3], 32.0 ^[4]
	(2S)-1-[(2S)-2-[[(2S)-2-Amino-2-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]-N-[(2S)-1-[[(2S)-1-[[1-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-6-methyl-1-oxoheptan-4-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide	Ki	10.0 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Renin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 Jul. 2026, https://www.aatbio.com/data-sets/renin-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2026, July 8). Quest Database™ Renin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/renin-inhibitors-ic50-ki.
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