X
Navigation Menu
Products
Services
Tools
Resources
logo
AAT Bioquest

 
search
logo
AAT Bioquest
Contact us
Company
Telephone:1-408-733-1055
Fax:1-408-733-1304
Hours:Monday to Friday
8:30 - 17:30 PST (GMT-8)
Location:5775 W Las Positas Blvd.
Pleasanton, CA, 94588
USA

Email us
Sales:sales@aatbio.com
Technical Support:support@aatbio.com
Website:websupport@aatbio.com
General Inquiries:info@aatbio.com
Order info
United States of America
Telephone:1-408-733-1055
Fax:1-408-733-1304
Email:sales@aatbio.com
Purchase Order:sales@aatbio.com

International
Click here to see all available distributors
Products
Services
Tools
Resources
 
search
calculatorCalculator

Retinoic acid receptor alpha Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
TretinoinIC500.78 [1], 0.89 [2], 15.0 [3], 9000.0 [4]
TretinoinKi0.1 [1], 3.3 [2], 16.0 [3], 187.0 [4]
BexaroteneKi180.0 [1], 1000.0 [2], 5453.0 [3]
AlitretinoinIC507.0 [1]
AlitretinoinKi22.3 [1]
AdapaleneKi1100.0 [1]
TamibaroteneIC5078.0 [1]
TamibaroteneKi6.5 [1]
TtnpbIC5036.0 [1]
TtnpbKi21.0 [1]
6-(1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopropyl)nicotinic acidKi1550.0 [1], 2745.0 [2]
(2E,4E,6Z)-7-[3,5-Ditert-butyl-2-(2,2-difluoroethoxy)phenyl]-3-methylocta-2,4,6-trienoic acidKi54.0 [1], 1000.0 [2]
6-(1,2,3,4-Tetrahydro-1,1,4,4-tetramethyl-6-naphthyl)-2-naphthalenecarboxylic acidKi580.0 [1]
6-(3-Tert-butyl-4-hydroxyphenyl)-2-naphthoic acidKi3000.0 [1], 10000.0 [2]
(E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzofuran-2-yl]prop-2-enoic acidIC501000.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-3-propoxy-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzofuran-2-yl]prop-2-enoic acidKi1000.0 [1]
6-[3-(1-Adamantyl)-4-hydroxyphenyl]-2-naphthalenecarboxylic AcidKi6500.0 [1]
4-{[(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)carbonyl]amino}benzoic acidIC5041.0 [1]
4-[2-[5,5-Dimethyl-8-(4-methylphenyl)-6H-naphthalen-2-yl]ethynyl]benzoic acidIC5031.0 [1]
4-(2,18,18,21,21-Pentamethyl-2,14-diazapentacyclo[13.8.0.03,12.04,9.017,22]tricosa-1(15),3(12),4,6,8,10,13,16,22-nonaen-13-yl)benzoic acidKi1300.0 [1]
4-(5,7,7,10,10-Pentamethyl-8,9-dihydronaphtho[2,3-b][1,4]benzodiazepin-13-yl)benzoic acidKi1400.0 [1]
(2E,4E,6Z)-3-Methyl-7-(5,5,8,8-tetramethyl-3-propoxy-6,7-dihydronaphthalen-2-yl)octa-2,4,6-trienoic acidKi1791.0 [1]
4-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-anthracenyl)benzoic acidKi5.3 [1]
4-{(E)-2-[5,5-Dimethyl-8-(phenylethynyl)-5,6-dihydronaphthalen-2-yl]ethenyl}benzoic acidIC50114.0 [1]
4-(7,7,10,10-Tetramethyl-8,9-dihydronaphtho[2,3-b][1,5]benzothiazepin-12-yl)benzoic acidKi900.0 [1]
6-(4-Methoxy-3-(1-methylcyclohexyl)phenyl)-2-naphthalenecarboxylic acidKi1120.0 [1]
7-(3,5-Ditert-butylphenyl)-3-methylocta-2,4,6-trienoic acidKi1.1 [1]
Benzoic acid, 4-(4-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-quinoxalinyl)-2-thiazolyl)-IC5083.0 [1]
6-[[3-[(2S)-1-Methoxypropan-2-yl]oxy-5-[(2S)-1-phenylpropan-2-yl]oxybenzoyl]amino]pyridine-3-carboxylic acidIC50470.0 [1]
4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalene-2-carbonyl)benzoic acidKi10000.0 [1]
4-[5-(4-Phenyl-8-propan-2-ylquinolin-2-yl)-1H-pyrrol-2-yl]benzoic acidIC5031.2 [1]
4-(2-(5,6,7,8-Tetrahydro-3,5,5,8,8-pentamethyl-2-naphthalenyl)-1-propenyl) benzoic acidIC50638.0 [1]
3-[(2S)-1-Methoxypropan-2-yl]oxy-5-(4-methylsulfonylphenoxy)-N-(3-methyl-1,2,4-thiadiazol-5-yl)benzamideIC5030000.0 [1]
4-{3-[3-Adamantan-1-yl-4-(2-methoxy-ethoxymethoxy)-phenyl]-3-oxo-propenyl}-benzoic acidIC504474.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-9-[2,6,6-trimethyl-3-(1,2,4-triazol-1-yl)cyclohexen-1-yl]nona-2,4,6,8-tetraenoic acidIC501000000.0 [1]
Benzoic acid, 4-(5-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-quinoxalinyl)-1H-pyrrol-2-yl)-IC502.2 [1]
4-((+/-)-(1H-Imidazol-1-yl)-(E)-retinoic acidIC5020000.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-9-[2,6,6-trimethyl-3-(1,2,4-triazol-4-yl)cyclohexen-1-yl]nona-2,4,6,8-tetraenoic acidIC50410000.0 [1]
4-[(5,5,8,8-Tetramethyl-6,7-dihydroquinoxaline-2-carbonyl)amino]benzoic acidIC5040.0 [1]
4-[(E)-2-(3-Tert-Butyl-4-methoxy-phenyl)-propenyl]-benzoic acidKi130.0 [1]
(S)-6-(3-(3,5-Difluorophenoxy)-5-(1-methoxypropan-2-yloxy)benzamido)nicotinic acidIC501.0 [1]
(2E,4E,6E)-7-[3,5-Ditert-butyl-2-(2,2-difluoroethoxy)phenyl]-6-fluoro-3-methylocta-2,4,6-trienoic acidKi8300.0 [1]
4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-vinyl]-benzoic acidKi944.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-5-(2-fluorophenyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi6756.0 [1]
4-[(E)-2-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-propenyl]-benzoic acidIC50100.0 [1]
6-(3-Isobutoxy-5-isopropoxy-benzoylamino)-nicotinic acidIC5010.0 [1]
(E)-3-[4-[3,5-Ditert-butyl-2-(3-fluoropropoxy)phenyl]-1-benzothiophen-2-yl]but-2-enoic acidKi7280.0 [1]
4-(7,7,10,10-Tetramethyl-8,9-dihydronaphtho[2,3-b][1,5]benzoxazepin-12-yl)benzoic acidKi980.0 [1]
4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-anthracen-2-yl)-benzoic acidIC5020.0 [1]
(E)-3-[4-(3,5,5,8,8-Pentamethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzofuran-2-yl]prop-2-enoic acidKi1000.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]prop-2-enoic acidKi1000.0 [1]
(E)-3-[4-(3,5-Diisopropyl-2-propoxy-phenyl)-benzo[b]thiophen-2-yl]-but-2-enoic acidKi6910.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1,3-benzoxazol-2-yl]prop-2-enoic acidKi1000.0 [1]
4-[5,5-Dimethyl-8-(5-methyl-2-thienyl)-5,6-dihydroanthracene-2-yl]benzoic acidIC5020.0 [1]
(E)-3-[7-(3,5-Diisopropyl-2-propoxy-phenyl)-benzofuran-2-yl]-but-2-enoic acidKi8500.0 [1]
6-[3-Adamantan-1-yl-4-(1,2-dihydroxy-ethyl)-phenyl]-naphthalene-2-carboxylic acidKi10000.0 [1]
(Z)-3-[7-[2-(2,2-Difluoroethoxy)-3,5-di(propan-2-yl)phenyl]-1-benzofuran-2-yl]-2-fluorobut-2-enoic acidKi10000.0 [1]
(E)-3-[4-[3,5-Ditert-butyl-2-(2,2-difluoroethoxy)phenyl]-1-benzothiophen-2-yl]but-2-enoic acidKi8360.0 [1]
(E)-3-[4-[3,5-Ditert-butyl-2-(3,3-difluoropropoxy)phenyl]-1-benzothiophen-2-yl]but-2-enoic acidKi10000.0 [1]
(E)-3-[4-[3,5-Ditert-butyl-2-(2,2,2-trifluoroethoxy)phenyl]-1-benzothiophen-2-yl]but-2-enoic acidKi10000.0 [1]
(E)-3-{7-[2-(3-Fluoro-propoxy)-3,5-diisopropyl-phenyl]-benzofuran-2-yl}-but-2-enoic acidKi10000.0 [1]
6-[3-Adamantan-1-yl-4-(2,3-dihydroxy-propoxy)-phenyl]-naphthalene-2-carboxylic acidKi5000.0 [1]
4-{(E)-4-[2-(4-Tert-Butyl-phenyl)-6,6-dimethyl-cyclohex-1-enyl]-but-3-en-1-ynyl}-benzoic acidIC50875.0 [1]
(E)-3-[4-(3-Methoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzofuran-2-yl]prop-2-enoic acidKi1000.0 [1]
(E)-3-[7-(2-Ethoxy-3,5-diisopropyl-phenyl)-benzo[b]thiophen-2-yl]-but-2-enoic acidKi6024.0 [1]
(E)-3-[4-(2-Ethoxy-3,5-diisopropyl-phenyl)-benzo[b]thiophen-2-yl]-but-2-enoic acidKi10000.0 [1]
(E)-3-[7-(2-Ethoxy-3,5-diisopropyl-phenyl)-benzofuran-2-yl]-but-2-enoic acidKi10000.0 [1]
(E)-3-[7-[2-(2,2-Difluoroethoxy)-3,5-di(propan-2-yl)phenyl]-1-benzofuran-2-yl]but-2-enoic acidKi10000.0 [1]
4-(8,8,11,11-Tetramethyl-10,13-dihydro-9H-naphtho[2,3-c][1]benzazepin-6-yl)benzoic acidKi1600.0 [1]
4-[(E)-2-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-propenyl]-benzoic acidIC501000.0 [1]
4-[(E)-4-(3,3-Dimethyl-6-p-tolyl-cyclohexa-1,5-dienyl)-but-3-en-1-ynyl]-benzoic acidIC50225.0 [1]
4-[(E)-2-(3-Adamantan-1-yl-4-hydroxy-phenyl)-propenyl]-benzoic acidKi1144.0 [1]
6-[3-(1-Adamantyl)-4-(2,3-dihydroxypropyl)phenyl]-2-naphthoic acidKi10000.0 [1]
4-(2,2-Dimethyl-4-p-tolyl-2H-1-thia-anthracen-6-yl)-benzoic acidIC501.5 [1]
4-[(E)-2-(3-Tert-butyl-4-hydroxyphenyl)propenyl]benzoic acidKi834.0 [1]
4-[(E)-2-[3-(1-Adamantyl)-4-hydroxyphenyl]ethenyl]benzoic acidKi610.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)thiophen-3-yl]benzoic acidIC502.4 [1]
4-(8,8,11,11,13-Pentamethyl-10,13-dihydro-9H-naphtho[2,3-c][1]benzazepin-6-yl)benzoic acidKi2000.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)furan-3-yl]benzoic acidIC5019.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)thiophen-2-yl]benzoic acidIC50130.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)furan-2-yl]benzoic acidIC5032.0 [1]
(2E,4E,6Z)-7-(3-Ethoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-3-methylocta-2,4,6-trienoic acidKi2582.0 [1]
4-{(E)-2-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-propenyl}-benzoic acidKi1056.0 [1]
4-[(E)-2-(3-(1-Methylcyclohexyl)-4-methoxyphenyl)propenyl]benzoic acidKi420.0 [1]
6-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-naphthalene-2-carboxylic acidKi10000.0 [1]
4-[(E)-2-(3-Adamantan-1-yl-4-methoxy-phenyl)-propenyl]-benzoic acidKi460.0 [1]
6-(3-Adamantan-1-yl-4-carboxy-phenyl)-naphthalene-2-carboxylic acidKi10000.0 [1]
6-[3-(1-Adamantyl)-4-(3-hydroxypropyl)phenyl]-2-naphthoic acidKi695.0 [1]
(E)-3-[5-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)furan-2-yl]prop-2-enoic acidKi93.0 [1]
3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]propanoic acidKi1000.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-1-(1,2,4-triazol-1-yl)-9-(2,6,6-trimethylcyclohexen-1-yl)nona-2,4,6,8-tetraen-1-oneIC5020000.0 [1]
(2Z,4E,6E,8E)-9-(3-Imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl)-3,7-dimethylnona-2,4,6,8-tetraenoic acidIC50100000.0 [1]
(E)-3-[6-Methyl-4-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-5,7-dihydro-4H-furo[2,3-c]pyridin-2-yl]prop-2-enoic acidKi1000.0 [1]
(2E,4E,6E,8E)-1-Imidazol-1-yl-3,7-dimethyl-9-(2,6,6-trimethylcyclohexen-1-yl)nona-2,4,6,8-tetraen-1-oneIC501000000.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-ylmethyl)-furan-2-yl]-acrylic acidKi1000.0 [1]
(E)-3-[5-Methyl-4-[(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)methyl]furan-2-yl]prop-2-enoic acidKi1000.0 [1]
(E)-3-[4-(5,5,8,8-Tetramethyl-6,7-dihydronaphthalen-2-yl)-4,5,6,7-tetrahydro-1-benzofuran-2-yl]but-2-enoic acidKi1000.0 [1]
(2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-3-methylocta-2,4,6-trienoic acidKi306.0 [1]
6-(3-Adamantan-1-yl-4-hexyloxy-phenyl)-naphthalene-2-carboxylic acidKi10000.0 [1]
4-[2-[5-(1-Adamantyl)-4-hydroxy-2-methylphenyl]-1,3-thiazol-5-yl]benzoic acidIC501277.0 [1]
Items per page: 1 - 10 of 100
⟨⟩

References

This online tool may be cited as follows

MLA

"Quest Database™ Retinoic acid receptor alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/retinoic-acid-receptor-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Retinoic acid receptor alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/retinoic-acid-receptor-alpha-inhibitors-ic50-ki.
BibTeXEndNoteRefMan
Location: Home / Datasets / Retinoic acid receptor alpha Inhibitors (IC50, Ki)
AboutPrivacyTerms of UseTerms of SalesDistributors
Copyright © 2024 AAT Bioquest, Inc. All Rights Reserved.