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Rho-associated protein kinase Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
N1-Benzyl-N4-(1H-5-indazolyl)-1,4-cyclohexanediamineIC50320.0 [1], 520.0 [2]
N1-Phenylethyl-N4-(5-isoquinolyl)-1,4-cyclohexanediamineIC50440.0 [1], 580.0 [2]
N1-Cyclopropyl-N4-(5-isoquinolyl)-1,4-cyclohexanediamineIC5070.0 [1], 195.0 [2]
N1-Propyl-N4-(5-isoquinolyl)-1,4-cyclohexanediamineIC50180.0 [1]
FasudilIC50180.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseRho-associated protein kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc.29 Dec2025https://www.aatbio.com/data-sets/rho-associated-protein-kinase-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 29). Quest DatabaseRho-associated protein kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/rho-associated-protein-kinase-inhibitors-ic50-ki.
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