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Secreted frizzled-related protein 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Tert-butyl (2S)-2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylateIC5060.0 [1]
5-(Phenylsulfonyl)-N-(1-L-prolylpiperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamideIC50110.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50200.0 [1]
Tert-butyl (2R)-2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylateIC50120.0 [1]
5-(Phenylsulfonyl)-N-(piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamideIC50500.0 [1]
5-(Benzenesulfonyl)-N-[1-(6-chloropyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50110.0 [1]
(2S)-2-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-N-tert-butylpyrrolidine-1-carboxamideIC5020.0 [1]
N-[1-(N-Methylglycyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)-benzenesulfonamideIC50200.0 [1]
N-[1-(N,N-Dimethylglycyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoro-methyl)benzenesulfonamideIC50300.0 [1]
N-[1-(Morpholin-4-ylacetyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC50100.0 [1]
5-(Benzenesulfonyl)-N-[1-(2-imidazol-1-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5030.0 [1]
Tert-butyl (2S)-2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-5-oxopyrrolidine-1-carboxylateIC50130.0 [1]
N-[1-[(2S)-1-Acetylpyrrolidine-2-carbonyl]piperidin-4-yl]-5-(benzenesulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC50160.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(2,2-dimethylpropanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-[2-(dimethylamino)acetyl]pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5090.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-benzoylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5070.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-[4-(dimethylamino)benzoyl]pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50110.0 [1]
(2S)-2-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-N-ethylpyrrolidine-1-carboxamideIC5030.0 [1]
(2S)-2-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-N-phenylpyrrolidine-1-carboxamideIC5020.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(morpholine-4-carbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(3,3-dimethylbutyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5030.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(cyclohexylmethyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
5-(Benzenesulfonyl)-N-[1-(2-pyrrolidin-1-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50110.0 [1]
5-(Phenylsulfonyl)-N-[1-(piperazin-1-ylacetyl)piperidin-4-yl]-2-(trifluoro-methyl)benzenesulfonamideIC50140.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-methylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50120.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-benzylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC501400.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-5-oxopyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5090.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(2-methylpropanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(3,3-dimethylbutanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5020.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(cyclohexanecarbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5050.0 [1]
5-(Benzenesulfonyl)-N-[1-[(2S)-1-(pyridine-4-carbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5070.0 [1]
(2S)-2-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-N,N-dimethylpyrrolidine-1-carboxamideIC5030.0 [1]
5-(Phenylsulfonyl)-N-[1-(piperidin-4-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50100.0 [1]
3-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]sulfonylbenzoic acidIC5020.0 [1]
5-(Benzenesulfonyl)-N-[1-[6-(dimethylamino)pyridine-3-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
N-[1-(4-Chlorobenzoyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC50300.0 [1]
5-(Benzenesulfonyl)-2-(trifluoromethyl)-N-[1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl]benzenesulfonamideIC50400.0 [1]
5-(Benzenesulfonyl)-N-[1-[4-(dimethylamino)benzoyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50300.0 [1]
5-(Phenylsulfonyl)-N-[1-(pyridin-2-ylcarbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50200.0 [1]
5-(Phenylsulfonyl)-N-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5060.0 [1]
N-(1-Isonicotinoylpiperidin-4-yl)-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC5080.0 [1]
5-(Benzenesulfonyl)-2-(trifluoromethyl)-N-[1-[6-(trifluoromethyl)pyridine-3-carbonyl]piperidin-4-yl]benzenesulfonamideIC5050.0 [1]
5-(Benzenesulfonyl)-N-[1-(6-pyrrolidin-1-ylpyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50870.0 [1]
5-(Benzenesulfonyl)-N-[1-(6-morpholin-4-ylpyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50130.0 [1]
Tert-butyl 4-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]piperidine-1-carboxylateIC50300.0 [1]
Tert-butyl 4-[2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]-2-oxoethyl]piperidine-1-carboxylateIC50490.0 [1]
Tert-butyl (3S)-3-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylateIC5070.0 [1]
Tert-butyl (3R)-3-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylateIC5050.0 [1]
5-(Benzenesulfonyl)-N-[1-(piperidine-4-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50120.0 [1]
5-(Benzenesulfonyl)-N-[1-[(3S)-pyrrolidine-3-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5040.0 [1]
5-(Benzenesulfonyl)-N-[1-[(3R)-pyrrolidine-3-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5060.0 [1]
2-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]acetamideIC5060.0 [1]
2-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]acetic acidIC50190.0 [1]
3-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]propanoic acidIC50900.0 [1]
4-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]-4-oxobutanoic acidIC50270.0 [1]
5-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]-5-oxopentanoic acidIC50500.0 [1]
5-(Benzenesulfonyl)-N-[1-(3-hydroxypropyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50500.0 [1]
5-(Benzenesulfonyl)-N-[1-(3-hydroxy-3-methylbutyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50200.0 [1]
5-(Phenylsulfonyl)-N-[1-(phenylsulfonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC50130.0 [1]
4-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]sulfonylbenzoic acidIC5020.0 [1]
5-(Benzenesulfonyl)-N-[1-(3-cyanophenyl)sulfonylpiperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5090.0 [1]
5-(Benzenesulfonyl)-N-[1-[3-(2H-tetrazol-5-yl)phenyl]sulfonylpiperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamideIC5030.0 [1]
3-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]benzoic acidIC50100.0 [1]
4-[4-[[5-(Benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]benzoic acidIC50120.0 [1]
5-(Benzenesulfonyl)-N-(1-benzoylpiperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamideIC5070.0 [1]
N-[1-(2-Chlorobenzoyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC50200.0 [1]
N-[1-(3-Chlorobenzoyl)piperidin-4-yl]-5-(phenylsulfonyl)-2-(trifluoromethyl)benzenesulfonamideIC50300.0 [1]
Items per page: 1 - 10 of 67
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References

This online tool may be cited as follows

MLA

"Quest Database™ Secreted frizzled-related protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/secreted-frizzled-related-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Secreted frizzled-related protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/secreted-frizzled-related-protein-1-inhibitors-ic50-ki.
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