Name: Serine protease hepsin Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Serine protease hepsin Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Nafamostat	IC50	5.0 ^[1]
	Nafamostat	Ki	0.53 ^[1]
	(2R)-N-(4-Carbamimidoylphenyl)-2-cyclohexyl-2-[(4-fluorophenyl)sulfonylamino]acetamide	IC50	90.0 ^[1], 190.0 ^[2], 1290.0 ^[3]
	(2R)-N-(4-Carbamimidoylphenyl)-2-cyclohexyl-2-[[4-(trifluoromethyl)phenyl]sulfonylamino]acetamide	IC50	680.0 ^[1], 850.0 ^[2], 3150.0 ^[3]
	(2R)-N-(4-Carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)sulfonylamino]acetamide	IC50	33.0 ^[1], 38.0 ^[2], 990.0 ^[3]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Serine protease hepsin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 6 Dec. 2025, https://www.aatbio.com/data-sets/serine-protease-hepsin-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 6). Quest Database™ Serine protease hepsin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-protease-hepsin-inhibitors-ic50-ki.
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