Serine/threonine-protein kinase 17A Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-[5-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]cyclohexanecarboxamide	IC50	1330.0 [1]
	Doramapimod	IC50	30000.0 [1]
	Sulfuretin	IC50	5850.0 [1]
	1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea	IC50	10.0 [1]
	Tomivosertib	IC50	131.0 [1]
	Chembl4126445	IC50	10.0 [1]
	1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid	IC50	10000.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2,2-dimethylpropanamide	IC50	32.0 [1]
	1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea	IC50	30000.0 [1]
	6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one	IC50	10000.0 [1]
	(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-one	IC50	12.8 [1]
	N-[2-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyrazin-7-yl]cyclohexanecarboxamide	IC50	4940.0 [1]
	Drak2-IN-1	IC50	51.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-nitrobenzamide	IC50	500.0 [1]
	4-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	780.0 [1]
	2-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	250.0 [1]
	4-Chloro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	3000.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	360.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclohexanecarboxamide	IC50	110.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclopropanecarboxamide	IC50	21.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-methylbut-2-enamide	IC50	120.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,3-dimethylbutanamide	IC50	24.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]butanamide	IC50	12.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]naphthalene-1-carboxamide	IC50	700.0 [1]
	(E)-N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-phenylprop-2-enamide	IC50	1100.0 [1]
	2-(3-Chlorophenoxy)-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]acetamide	IC50	460.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2-(trifluoromethyl)benzamide	IC50	320.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methoxybenzamide	IC50	360.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methylbenzamide	IC50	1300.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,5-dinitrobenzamide	IC50	24.0 [1]
	(2Z)-2-[(3,4-Dihydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one	IC50	5810.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one	IC50	1410.0 [1]
	N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2,2-dimethylbutanamide	IC50	2100.0 [1]
	(2R)-N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2-methylbutanamide	IC50	2900.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 34 ⟨⟩

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ Serine/threonine-protein kinase 17A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17a-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Serine/threonine-protein kinase 17A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17a-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan