Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-[5-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]cyclohexanecarboxamide	IC50	720.0 [1]
	Drak2-IN-1	IC50	3.0 [1]
	Drak2-IN-1	Ki	0.26 [1]
	Staurosporine	IC50	25.8 [1]
	Indirubin	IC50	10000.0 [1]
	Indirubin-3'-monoxime	IC50	710.0 [1]
	Aurone	IC50	24640.0 [1]
	Sulfuretin	IC50	1020.0 [1]
	3-(1,3-Dihydro-3-oxo-2H-indol-2-ylidene)-1,3-dihydro-5-iodo-2H-indol-2-one	IC50	6200.0 [1]
	5'-Fluoroindirubinoxime	IC50	620.0 [1]
	(3Z)-5-Methyl-3-(3-oxoindolin-2-ylidene)indolin-2-one	IC50	10000.0 [1]
	(3Z)-5-Fluoro-3-(3-oxoindolin-2-ylidene)indolin-2-one	IC50	10000.0 [1]
	(3Z)-5-Chloro-3-(3-oxoindolin-2-ylidene)indolin-2-one	IC50	10000.0 [1]
	(Z)-2-(3,4-Dimethoxybenzylidene)benzofuran-3(2H)-one	IC50	21430.0 [1]
	2-(4-Hydroxybenzylidene)-1-benzofuran-3(2H)-one	IC50	53030.0 [1]
	2-[(Z)-3,4-Dihydroxybenzylidene]-2,3-dihydrobenzofuran-3-one	IC50	3080.0 [1]
	2-(3,4-Dihydroxybenzylidene)indan-1-one	IC50	13290.0 [1]
	2-(5-Amino-2-hydroxy-1H-indol-3-yl)indol-3-one	IC50	1400.0 [1]
	5-Amino-3-(3-nitroso-1H-indol-2-yl)-1H-indol-2-ol	IC50	250.0 [1]
	2-(4-Fluorobenzylidene)benzofuran-3(2H)-one	IC50	40550.0 [1]
	2-[(Z)-3-Methoxy-4-hydroxybenzylidene]-2,3-dihydrobenzofuran-3-one	IC50	3110.0 [1]
	(2Z)-2-[(3-Hydroxy-4-methoxyphenyl)methylidene]-1-benzofuran-3-one	IC50	12100.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2,2-dimethylpropanamide	IC50	21.0 [1]
	5-Chloro-7-methyl-3-(3-nitroso-1H-indol-2-yl)-1H-indol-2-ol	IC50	10000.0 [1]
	2-[(Z)-3-Ethoxy-4-hydroxybenzylidene]-2,3-dihydrobenzofuran-3-one	IC50	3240.0 [1]
	5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide	IC50	10000.0 [1]
	(2Z)-2-(Pyridin-3-ylmethylidene)-1-benzofuran-3-one	IC50	39390.0 [1]
	Sulferetol	IC50	990.0 [1]
	N-[2-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyrazin-7-yl]cyclohexanecarboxamide	IC50	1780.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-nitrobenzamide	IC50	1300.0 [1]
	4-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	1200.0 [1]
	2-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	290.0 [1]
	4-Chloro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	3200.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide	IC50	200.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclohexanecarboxamide	IC50	120.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclopropanecarboxamide	IC50	8.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-methylbut-2-enamide	IC50	14.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,3-dimethylbutanamide	IC50	14.0 [1]
	4-Bromo-2-(2-hydroxy-5-nitro-1H-indol-3-yl)indol-3-one	IC50	10000.0 [1]
	2-(5-Chloro-2-hydroxy-7-methyl-1H-indol-3-yl)indol-3-one	IC50	10000.0 [1]
	2-(2-Hydroxy-5,7-dimethyl-1H-indol-3-yl)indol-3-one	IC50	10000.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]butanamide	IC50	10.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]naphthalene-1-carboxamide	IC50	1500.0 [1]
	(E)-N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-phenylprop-2-enamide	IC50	700.0 [1]
	2-(3-Chlorophenoxy)-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]acetamide	IC50	950.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2-(trifluoromethyl)benzamide	IC50	120.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methoxybenzamide	IC50	330.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methylbenzamide	IC50	1300.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,5-dinitrobenzamide	IC50	77.0 [1]
	4-Bromo-2-(2-hydroxy-1H-indol-3-yl)indol-3-one	IC50	10000.0 [1]
	2-[(3,4-Dihydroxyphenyl)methyl]-1-benzofuran-3-one	IC50	27810.0 [1]
	5-(3-Amino-5-thiophen-3-ylthieno[2,3-b]pyridin-2-yl)-3H-1,3,4-oxadiazole-2-thione	IC50	29.0 [1]
	(2Z)-2-[[4-(Hydroxymethyl)phenyl]methylidene]-1-benzofuran-3-one	IC50	11090.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-fluoro-1-benzofuran-3-one	IC50	1050.0 [1]
	(2Z)-5-Butoxy-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	3660.0 [1]
	(2Z)-2-[(3,4-Dihydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one	IC50	250.0 [1]
	(2Z)-6-Chloro-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	40540.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-iodo-1-benzofuran-3-one	IC50	42520.0 [1]
	(2Z)-2-[(4-Hydroxy-3-propan-2-yloxyphenyl)methylidene]-1-benzofuran-3-one	IC50	17390.0 [1]
	(2Z)-5-Ethoxy-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	410.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-7-methoxy-1-benzofuran-3-one	IC50	1290.0 [1]
	(2Z)-2-[(4-Hydroxy-3,5-dimethoxyphenyl)methylidene]-1-benzofuran-3-one	IC50	6650.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-4-methoxy-1-benzofuran-3-one	IC50	7260.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one	IC50	330.0 [1]
	(2Z)-5-Amino-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	7160.0 [1]
	1-Benzofuran-2-yl-(3,4-dihydroxyphenyl)methanone	IC50	22910.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-6-fluoro-1-benzofuran-3-one	IC50	60400.0 [1]
	(2Z)-2-[(3-Butoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	29100.0 [1]
	[(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-3-oxo-1-benzofuran-5-yl] acetate	IC50	690.0 [1]
	(2Z)-2-[(4-Hydroxy-3-propoxyphenyl)methylidene]-1-benzofuran-3-one	IC50	5370.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-6-methoxy-1-benzofuran-3-one	IC50	2440.0 [1]
	(2Z)-5-Bromo-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	28150.0 [1]
	(2Z)-5-Chloro-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-one	IC50	13710.0 [1]
	(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methyl-1-benzofuran-3-one	IC50	960.0 [1]
	(2Z)-2-Furfurylidenebenzofuran-3(2H)-one	IC50	63960.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 75 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17b-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17b-inhibitors-ic50-ki.
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