Name: Serine/threonine-protein kinase PLK1 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Serine/threonine-protein kinase PLK1 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	BI-2536	IC50	0.83 ^[1]
	BI-2536	Ki	0.22 ^[1], 3.0 ^[2]
	[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-(8-phenyloctyl)imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate	IC50	25.0 ^[1]
	Staurosporine	IC50	540.0 ^[1]
	[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate	IC50	300.0 ^[1], 16000.0 ^[2], 21500.0 ^[3], 300000.0 ^[4]
Rows per page: 1–5 of 100

References

This online resource may be cited as follows

MLA	"Quest Database™ Serine/threonine-protein kinase PLK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 14 Dec. 2025, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 14). Quest Database™ Serine/threonine-protein kinase PLK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk1-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan