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Serine/threonine-protein kinase PLK4 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
AxitinibIC5043.0 [1], 46.0 [2]
AxitinibKi4.2 [1]
CFI-400945 (free base)IC502.8 [1]
CFI-400945 (free base)Ki0.26 [1]
3-[(E)-[3-[(E)-2-[4-[(Dimethylamino)methyl]phenyl]ethenyl]indazol-6-ylidene]methyl]-1H-indol-2-olIC502.0 [1], 4.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerine/threonine-protein kinase PLK4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk4-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseSerine/threonine-protein kinase PLK4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk4-inhibitors-ic50-ki.
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