Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Axitinib | IC50 | 43.0 [1], 46.0 [2] | |
| Axitinib | Ki | 4.2 [1] | |
| CFI-400945 (free base) | IC50 | 2.8 [1] | |
| CFI-400945 (free base) | Ki | 0.26 [1] | |
| 3-[(E)-[3-[(E)-2-[4-[(Dimethylamino)methyl]phenyl]ethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 2.0 [1], 4.0 [2] | |
MLA | "Quest Database™ Serine/threonine-protein kinase PLK4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk4-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Serine/threonine-protein kinase PLK4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-plk4-inhibitors-ic50-ki. | |
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