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Serine/threonine-protein kinase Sgk1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Sgk1-IN-1IC501.0 [1]
N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2,3-dichlorobenzenesulfonamideIC503.0 [1]
Sgk1-IN-2IC505.0 [1], 25.0 [2], 630.0 [3]
N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluorophenyl]-5-chloro-2-fluorobenzenesulfonamideIC502.0 [1], 50.0 [2], 2100.0 [3]
N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluorophenyl]-2,5-dichlorobenzenesulfonamideIC502.0 [1], 13.0 [2], 2600.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerine/threonine-protein kinase Sgk1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-sgk1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseSerine/threonine-protein kinase Sgk1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-sgk1-inhibitors-ic50-ki.
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