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Serine/threonine-protein kinase ULK1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
CID 44464263IC502.9 [1], 170.0 [2]
N~2~-(1h-Benzimidazol-6-Yl)-N~4~-(5-Cyclobutyl-1h-Pyrazol-3-Yl)quinazoline-2,4-DiamineIC505.3 [1], 8.0 [2]
4-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamideIC501490.0 [1], 13960.0 [2]
CID 10077147IC5087.0 [1]
CID 92044402IC50108.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
N-[3-[[4-[3-(Cyclopropanecarbonylamino)propylamino]-5-iodopyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamideIC5067.0 [1]
Clk1-IN-1IC5010000.0 [1]
(1S,3R)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC503050.0 [1]
(1S,3R)-3-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamideIC50330.0 [1]
N-(3-Amino-1H-indazol-5-yl)piperidine-4-carboxamideIC50560.0 [1]
3-(Dimethylamino)-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC504230.0 [1]
N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]azetidine-3-carboxamideIC504940.0 [1]
3-Amino-N-[3-(2-fluoroanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50840.0 [1]
3-Hydroxy-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC502220.0 [1]
3-Amino-N-(3-anilino-1H-indazol-5-yl)cyclohexane-1-carboxamideIC502730.0 [1]
4-Amino-N-(3-amino-1H-indazol-5-yl)butanamideIC5033000.0 [1]
3-Amino-N-[3-(2-methoxyanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50110.0 [1]
3-Amino-N-(3-amino-1H-indazol-5-yl)benzamideIC5018100.0 [1]
3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC5011.0 [1]
Methyl 3-[[5-[(3-aminocyclohexanecarbonyl)amino]-1H-indazol-3-yl]amino]benzoateIC50183.0 [1]
3-Amino-N-[3-(quinolin-8-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50589.0 [1]
N-(3-Amino-1H-indazol-5-yl)piperidine-3-carboxamideIC50670.0 [1]
(1R,3S)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC5045.0 [1]
N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]oxane-4-carboxamideIC501830.0 [1]
3-Amino-N-[3-(quinolin-4-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50239.0 [1]
N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]piperidine-4-carboxamideIC50315.0 [1]
(1R,3R)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC5024.0 [1]
3-Amino-N-[3-[(4-methoxyphenyl)methylamino]-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50477.0 [1]
3-Amino-N-[3-[3-(trifluoromethyl)anilino]-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50288.0 [1]
N-[5-[(3-Aminocyclohexanecarbonyl)amino]-1H-indazol-3-yl]benzamideIC50242.0 [1]
N'-[3-[[5-Cyclopropyl-2-[(2-methyl-3,4-dihydro-1H-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboximidamideIC5045.0 [1]
N-(3-Amino-1H-indazol-5-yl)piperidine-2-carboxamideIC50840.0 [1]
3-Amino-N-[3-(4-bromoanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC50416.0 [1]
3-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamideIC50368.0 [1]
3-Amino-N-[3-(quinolin-5-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamideIC5040.0 [1]
3-Amino-N-(1H-indazol-5-yl)cyclohexane-1-carboxamideIC5022400.0 [1]
N-[3-({4-[(3-Aminopropyl)amino]-5-Iodopyrimidin-2-Yl}amino)phenyl]pyrrolidine-1-CarboxamideIC50120.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase ULK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-ulk1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Serine/threonine-protein kinase ULK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-ulk1-inhibitors-ic50-ki.
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