Serine/threonine protein phosphatase PP1-gamma catalytic subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Okadaic acid	IC50	260.0 [1]
	Microcystin-LR	IC50	0.8 [1]
	Calyculin A	IC50	48.0 [1]
	Cantharidin	IC50	1780.0 [1]
	4,7-Epoxyisobenzofuran-1,3-dione, hexahydro-, (3aR,4S,7R,7aS)-rel-	IC50	1980.0 [1]
	Tautomycetin	IC50	1.6 [1]
	(1R,2S,6R,7S)-5-Ethoxy-4,10-dioxatricyclo[5.2.1.02,6]decan-3-one	IC50	746000.0 [1]
	(1R,2S,6R,7S)-5-Propoxy-4,10-dioxatricyclo[5.2.1.02,6]decan-3-one	IC50	1000000.0 [1]
	(1R,2S,6R,7S)-5-Methoxy-4,10-dioxatricyclo[5.2.1.02,6]decan-3-one	IC50	1000000.0 [1]
	2-(4-(7-(4-Methoxybenzoyl)cyclopenta[d][1,2]oxazin-4-yl)phenoxy)acetic acid	IC50	35200.0 [1]
	7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid monopropyl ester	IC50	4820.0 [1]
	7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid monoethyl ester	IC50	2960.0 [1]
	7-Oxa-bicyclo[2.2.1]heptane-2,3-dicarboxylic acid monomethyl ester	IC50	4710.0 [1]
	2-(4-(7-(4-Tetradecylbenzoyl)cyclopenta[d][1,2]oxazin-4-yl)phenoxy)acetic acid	IC50	220.0 [1]
	2-[4-[7-[4-(Aminomethyl)benzoyl]cyclopenta[d]oxazin-4-yl]phenoxy]acetic acid	IC50	1300.0 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4E)-4-[2-(3-Benzoylanilino)-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	8.0 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4Z)-4-[2-(3-Benzoylanilino)-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	32.5 [1]
	Tautomycin diacid	Ki	4.5 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4E)-4-[2-[2-[2-[(3-Azido-4-fluorobenzoyl)amino]ethyldisulfanyl]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	19.6 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4Z)-4-[2-[2-[2-[(3-Azido-4-fluorobenzoyl)amino]ethyldisulfanyl]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	23.9 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4E)-4-[2-[3-[(3-Azido-4-fluorobenzoyl)amino]propylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	3.4 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4E)-4-[2-[2-[(3-Azido-4-fluorobenzoyl)amino]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	17.3 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-12-[(2S,3S,6R,8S,9R)-8-[(3S,4Z)-4-[2-[2-[(3-Azido-4-fluorobenzoyl)amino]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-5,9-dihydroxy-4-methoxy-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	8.4 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-5,9-Dihydroxy-4-methoxy-12-[(2S,3S,6R,8S,9R)-8-[(3S,4E)-4-[2-[2-[[2-methoxy-4-[3-(trifluoromethyl)diazirin-3-yl]benzoyl]amino]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	21.3 [1]
	(Z)-2-[(1R)-3-[(3R,4S,5R,8S,9S,12R)-5,9-Dihydroxy-4-methoxy-12-[(2S,3S,6R,8S,9R)-8-[(3S,4Z)-4-[2-[2-[[2-methoxy-4-[3-(trifluoromethyl)diazirin-3-yl]benzoyl]amino]ethylamino]-2-oxoethoxy]imino-3-methylpentyl]-3,9-dimethyl-1,7-dioxaspiro[5.5]undecan-2-yl]-2,8-dimethyl-7-oxotridecan-3-yl]oxy-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid	Ki	49.7 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 25 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Serine/threonine protein phosphatase PP1-gamma catalytic subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-phosphatase-pp1-gamma-catalytic-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Serine/threonine protein phosphatase PP1-gamma catalytic subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-phosphatase-pp1-gamma-catalytic-subunit-inhibitors-ic50-ki.
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