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Serotonin 1a (5-HT1a) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
8-OH-DpatIC500.59 [1], 0.66 [2]
8-OH-DpatKi0.4 [1]
SerotoninIC501.2 [1], 2.0 [2], 5.6 [3], 6.0 [4]
SerotoninKi2.48 [1], 2.8 [2], 3.0 [3]
BuspironeIC5025.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 1a (5-HT1a) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/serotonin-1a-5-ht1a-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseSerotonin 1a (5-HT1a) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-1a-5-ht1a-receptor-inhibitors-ic50-ki.
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