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Serotonin 1b (5-HT1b) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
SumatriptanKi23.1 [1]
SerotoninIC505.0 [1], 6.5 [2], 12.0 [3], 16.0 [4]
SerotoninKi6.76 [1]
6-((1-(2-((2-Methylquinolin-5-yl)oxy)ethyl)piperidin-4-yl)methyl)-2H-1,4-benzoxazin-3(4H)-oneKi10.0 [1]
6-[2-[4-(2-Methylquinolin-5-yl)piperazin-1-yl]ethyl]-4H-1,4-benzoxazin-3-oneKi0.2 [1], 0.5 [2], 251.19 [3]

References
This online resource may be cited as follows
MLA
"Quest Database™ Serotonin 1b (5-HT1b) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Oct. 2026, https://www.aatbio.com/data-sets/serotonin-1b-5-ht1b-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026, October 15). Quest Database™ Serotonin 1b (5-HT1b) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-1b-5-ht1b-receptor-inhibitors-ic50-ki.
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