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Serotonin 1f (5-HT1f) receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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4-Fluoro-N-[3-(1-methylpiperidin-4-yl)-1H-indol-5-yl]benzamideKi1.6 [1], 2.1 [2]
SumatriptanIC501000.0 [1]
SumatriptanKi25.7 [1]
5-Chloro-N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-3-methyl-1-benzothiophene-2-sulfonamideKi251.19 [1]
4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi7.6 [1]
(R)-3-((2-(2-(4-Methylpiperidin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)phenolKi3162.28 [1]
SB 224289Ki10000.0 [1]
5-Chloro-N-(4-methoxy-3-(piperazin-1-yl)phenyl)-3-methylbenzo[b]thiophene-2-sulfonamideKi1000.0 [1]
2-[1-(Benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamineKi2500.0 [1]
N,3-Dimethyl-N-[(2R)-4-(4-methylpiperidin-1-yl)butan-2-yl]benzenesulfonamideKi6309.57 [1]
1-(3-(5-(1,2,4-Triazol-4-yl)-1H-indol-3-yl)propyl)-4-(2-(3-fluorophenyl)ethyl)piperazineIC503800.0 [1]
N-(2,5-Dibromo-3-fluorophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamideKi10000.0 [1]
4-Methyl-1-[2-[(2R)-1-(3-methylphenyl)sulfonylpyrrolidin-2-yl]ethyl]piperidineKi10000.0 [1]
[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimethyl-amineKi770.0 [1]
CID 10028436Ki1995.26 [1]
CID 10436045Ki3.16 [1]
CID 9847194IC5010000.0 [1]
4-Bromo-N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]benzenesulfonamideKi316.23 [1]
1-(Phenylsulfonyl)-4-[2-(dimethylamino)ethyl]-1H-indoleKi3.9 [1]
N-[3-[(8As)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-4-methoxyphenyl]-5-chloro-3-methyl-1-benzothiophene-2-sulfonamideKi316.23 [1]
(2R)-1-(1-Naphthylsulfonyl)-2-[2-(4-methylpiperidino)ethyl]pyrrolidineKi10000.0 [1]
2-Methyl-5-(2-(4-(quinolin-8-ylmethyl)piperazin-1-yl)ethoxy)quinolineKi1995.26 [1]
N-(3-(1-(2-(2-Methylquinolin-5-yloxy)ethyl)piperidin-4-ylmethyl)phenyl)methanesulfonamideKi501.19 [1]
6-Iodo-1-indolinyl 3-piperazino-4-methoxyphenyl sulfoneKi7943.28 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-acetamideKi5.0 [1]
3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic acid ethyl esterKi2000.0 [1]
Benzamide,N-[(3S)-1-[[3-bromo-4-(4-piperidinyloxy)phenyl]methyl]-3-pyrrolidinyl]-3,4-dichloro-Ki7200.0 [1]
1-(2-Iodophenyl)-N-[3-[[(2R)-pyrrolidin-2-yl]methyl]-1H-indol-5-yl]methanesulfonamideKi17.8 [1]
7-[2-[2-(3-Chlorophenyl)ethylamino]ethyl]quinolin-2-AmineKi100.0 [1]
N-[3-(2-Dimethylamino-ethyl)-2-methyl-1H-indol-5-yl]-4-fluoro-benzamideKi8.2 [1]
4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-furo[3,2-b]pyridin-5-yl]-benzamideKi3.1 [1]
2-[2-[4-(5-Fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-4,5-dihydro-3H-2-benzazepin-1-oneKi10000.0 [1]
N-[3-[(8Ar)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-4-methoxyphenyl]-5-chloro-3-methyl-1-benzothiophene-2-sulfonamideKi199.53 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-propionamideKi5.5 [1]
2,4,6-Trifluoro-N-[3-(1-methyl-piperidin-4-yl)-furo[3,2-b]pyridin-5-yl]-benzamideKi2.3 [1]
5-Methoxy-3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridineKi23.0 [1]
3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-ylamineKi100.0 [1]
3-(1-Methyl-piperidin-4-yl)-1,4-dihydro-pyrrolo[3,2-b]pyridin-5-oneKi100.0 [1]
(E)-3-(3,4-Dichlorophenyl)-N-[4-[[(1R,5S)-3-(5-hydroxy-1H-indol-3-yl)-8-azabicyclo[3.2.1]octan-8-yl]methyl]cyclohexyl]prop-2-enamideKi3162.28 [1]
4-Fluoro-N-[6-(1-methylpiperidine-4-carbonyl)pyridin-2-yl]benzamideKi9.5 [1]
N-(2,5-Dibromophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamideKi10000.0 [1]
4-Methoxy-3-piperazin-1-yl-N-(2,3,5-trichlorophenyl)benzenesulfonamideKi10000.0 [1]
(2R)-1-(3-Bromophenylsulfonyl)-2-[2-(4-methylpiperidino)ethyl]pyrrolidineKi5011.87 [1]
(2R)-1-(1-Naphthylsulfonyl)-2-[2-(4-methylpiperidino)ethyl]piperidineKi10000.0 [1]
(2R)-1-(3,4-Dichlorophenylsulfonyl)-2-[2-(4-methylpiperidino)ethyl]pyrrolidineKi3162.28 [1]
4-Fluoro-N-[3-(1-isopropyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi30.0 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-4-nitro-benzamideKi7.7 [1]
4-Fluoro-N-[3-(1-phenethyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi75.0 [1]
N-[3-(1-Ethyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-acetamideKi21.0 [1]
N-[7-(1-Methylpiperidin-4-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-yl]acetamideKi220.0 [1]
4-Fluoro-N-[3-(1-methylpiperidin-4-yl)-1H-pyrrolo[2,3-c]pyridin-5-yl]benzamideKi13.0 [1]
3-Cyano-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi11.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]pentanamideKi14.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]furan-2-carboxamideKi13.0 [1]
3-Methyl-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi5.8 [1]
N-(3-Piperidin-4-yl-1H-pyrrolo[3,2-b]pyridin-5-yl)-acetamideKi45.0 [1]
N-(3-Piperidin-4-yl-1H-pyrrolo[3,2-b]pyridin-5-yl)-propionamideKi35.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]cyclobutanecarboxamideKi8.7 [1]
4-Fluoro-N-[3-(1-propyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi18.0 [1]
1-(4-Fluoro-phenyl)-3-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-ureaKi11.0 [1]
2,4-Dichloro-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi4.1 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]hexanamideKi13.0 [1]
N-[3-(2-Dimethylamino-ethyl)-2-methyl-furo[3,2-b]pyridin-5-yl]-4-fluoro-benzamideKi13.5 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-2-nitro-benzamideKi19.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]cyclopropanecarboxamideKi9.8 [1]
N-[3-(1-Ethyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-4-fluoro-benzamideKi25.0 [1]
4-Fluoro-N-[7-(1-methylpiperidin-4-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-yl]benzamideKi67.0 [1]
2-Methyl-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi12.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[2,3-c]pyridin-5-yl]acetamideKi210.0 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-butyramideKi6.9 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]thiophene-3-carboxamideKi7.4 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-3-nitro-benzamideKi42.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]thiophene-2-carboxamideKi7.1 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi7.3 [1]
4-Methyl-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi12.0 [1]
3-Methoxy-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi16.0 [1]
N-[3-(1-Butyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-4-fluoro-benzamideKi14.0 [1]
1-Methyl-3-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-ureaKi2.5 [1]
4-Fluoro-N-(3-piperidin-4-yl-1H-pyrrolo[3,2-b]pyridin-5-yl)-benzamideKi9.5 [1]
[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl] 4-fluorobenzenesulfonateKi7.5 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]pyridine-2-carboxamideKi6.3 [1]
2-Methoxy-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi20.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]furan-3-carboxamideKi4.6 [1]
2-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi19.0 [1]
N-[3-(1-Ethyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-4-fluoro-benzamideKi170.0 [1]
2,2-Dimethyl-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-propionamideKi62.0 [1]
2-Chloro-N-[3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indol-5-yl]benzenesulfonamideKi16.0 [1]
2-Chloro-N-[3-[[(2R)-pyrrolidin-2-yl]methyl]-1H-indol-5-yl]benzenesulfonamideKi12.3 [1]
2-Chloro-4-fluoro-N-[3-(1-methylpiperidin-4-yl)-1,2-benzoxazol-5-yl]benzamideKi3.6 [1]
3-Chloro-N-[3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indol-5-yl]benzenesulfonamideKi2.7 [1]
1-[2-Hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanoneKi2970000.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]cyclopentanecarboxamideKi11.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]octanamideKi20.0 [1]
N-[3-(1-Methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-isonicotinamideKi8.4 [1]
4-Fluoro-N-[3-(1-methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]benzenesulfonamideKi27.0 [1]
1-Ethyl-3-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-ureaKi3.8 [1]
[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl] methanesulfonateKi4.7 [1]
3-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]-benzamideKi11.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]methanesulfonamideKi19.0 [1]
N-[3-(1-Methylpiperidin-4-yl)-1H-pyrrolo[3,2-b]pyridin-5-yl]cyclohexanecarboxamideKi20.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serotonin 1f (5-HT1f) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/serotonin-1f-5-ht1f-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Serotonin 1f (5-HT1f) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-1f-5-ht1f-receptor-inhibitors-ic50-ki.
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