X
Navigation Menu
Products
Services
Tools
Resources
logo
AAT Bioquest

 
search
logo
AAT Bioquest
Contact us
Company
Telephone:1-408-733-1055
Fax:1-408-733-1304
Hours:Monday to Friday
8:30 - 17:30 PST (GMT-8)
Location:5775 W Las Positas Blvd.
Pleasanton, CA, 94588
USA

Email us
Sales:sales@aatbio.com
Technical Support:support@aatbio.com
Website:websupport@aatbio.com
General Inquiries:info@aatbio.com
Order info
United States of America
Telephone:1-408-733-1055
Fax:1-408-733-1304
Email:sales@aatbio.com
Purchase Order:sales@aatbio.com

International
Click here to see all available distributors
Products
Services
Tools
Resources
 
search
calculatorCalculator

Serotonin 2 (5-HT2) receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
HaloperidolKi16.0 [1], 19.95 [2], 34.0 [3]
2-Naphthalenecarboxamide, N-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-Ki840.0 [1]
ClozapineKi5.01 [1], 12.0 [2]
CisaprideIC506.1 [1]
3-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo[2,3-b]pyridineKi200.0 [1], 1000.0 [2]
4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochlorideIC5010000.0 [1]
4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochlorideKi10000.0 [1]
4-Amino-N-[(4R)-1-azatricyclo[3.3.1.03,7]nonan-4-yl]-5-chloro-2-methoxybenzamideIC5010000.0 [1]
OlanzapineKi10.0 [1]
QuetiapineKi220.0 [1]
8-OH-DpatKi1614.0 [1]
ZafirlukastIC5010000.0 [1]
RimcazoleKi2482.0 [1]
DR-4004Ki98.0 [1]
N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamideKi2000.0 [1]
1'-Benzyl-3,4-dihydro-2H-spiro[naphthalene-1,4'-piperidine]Ki1934.0 [1]
N-DesmethylolanzapineKi23.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamideKi1200.0 [1]
N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamideKi350.0 [1]
N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamideKi660.0 [1]
N-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamideKi11000.0 [1]
SpipethianeKi7600.0 [1]
DUP-734 free baseKi15.0 [1]
(1S,13R)-1,13-Dimethyl-10-prop-2-enyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
3-Propyl-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indol-9-olKi1637.0 [1]
2a-[3-(4-Phenylpiperazin-1-yl)propyl]-1,3,4,5-tetrahydrobenzo[cd]indol-2-oneKi16.0 [1]
N-((Hexahydro-1H-pyrrolizin-1-yl)methyl)-6-chloroimidazo(1,2-a)pyridine-8-carboxamide hydrochlorideIC5010000.0 [1]
2-Hydroxymethyl OlanzapineKi18.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-4-carboxamideKi1600.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-7-carboxamideKi2000.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-5-carboxamideKi740.0 [1]
N-Methyl-2-[2-[4-(2-oxo-1,3,4,5-tetrahydrobenzo[cd]indol-2a-yl)butyl]-3,4-dihydro-1H-pyrido[3,4-b]indol-9-yl]acetamideKi1000.0 [1]
2-(2-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-yl}-ethoxy)-benzoic acidIC5010000.0 [1]
3-{4-[1-(5-Chloro-thiophen-2-ylmethyl)-1H-indol-3-yl]-piperidin-1-ylmethyl}-benzoic acidIC5010000.0 [1]
1-[4-(Acetylaminomethyl)benzyl]-4-(2,4-difluorophenyl)piperazineKi1000.0 [1]
6-Chloro-1'-(2-phenylethyl)spiro[3,4-dihydronaphthalene-2,4'-piperidine]-1-oneKi119.0 [1]
5-{4-[1-(2-Ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}-2-methoxybenzoic acidIC5010000.0 [1]
1'-Benzylspiro[3,4-dihydrochromene-2,4'-piperidine]Ki10000.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-6-carboxamideKi950.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-3-carboxamideKi1300.0 [1]
2-(2-{4-[1-(2-Ethoxy-ethyl)-1H-indol-3-yl]-piperidin-1-yl}-ethoxy)-benzoic acidIC5010000.0 [1]
2-(2-{4-[1-(2-Ethoxyethyl)-1H-indol-3-yl]piperidin-1-yl}ethoxy)-4-methoxybenzoic acidIC503900.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]tricyclo[8.2.2.24,7]hexadeca-1(13),4,6,10(14),11,15-hexaene-5-carboxamideKi2300.0 [1]
1-[4-(Acetylaminomethyl)benzyl]-4-phenylpiperazineKi1000.0 [1]
5'-Chloro-N,N-dimethylspiro[cyclohex-2-ene-4,2'-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaene]-1-amineKi1.3 [1]
5'-Chloro-N,N-dimethylspiro[cyclohex-2-ene-4,2'-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene]-1-amineKi30.0 [1]
1'-(2-Phenylethyl)spiro[3,4-dihydro-1H-naphthalene-2,4'-piperidine]-1-olKi4.2 [1]
2-{2-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-benzoic acidIC5010000.0 [1]
4-{4-[1-(2-Ethoxyethyl)-1H-indol-3-yl]piperidin-1-ylmethyl}benzoic acidIC504950.0 [1]
19-Methoxy-5-methyl-2,5-diazatetracyclo[13.4.0.02,7.08,13]nonadeca-1(15),8,10,12,16,18-hexaeneKi56.0 [1]
2-[1-(4-Tert-Butylbenzyl)-4-piperidinyl]-3,4-dihydronaphthalen-1(2H)-oneKi176.0 [1]
N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-benzotellurophene-2-carboxamideKi730.0 [1]
6-Methoxy-2-[1-benzyl-4-piperidinyl]-3,4-dihydronaphthalen-1(2H)-oneKi282.0 [1]
6-Methoxy-2-[1-phenethyl-4-piperidinyl]-3,4-dihydronaphthalen-1(2H)-oneKi7.0 [1]
5-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-2-methoxy-benzoic acidIC5010000.0 [1]
2-{2-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-yl]-ethoxy}-benzoic acidIC5010000.0 [1]
(1R,9S,13S)-1,13-Dimethyl-10-(2-piperidin-1-ylethyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
6-Fluoro-2-[1-benzyl-4-piperidinyl]-3,4-dihydronaphthalen-1(2H)-oneKi101.0 [1]
1-[4-[2-Methylphenyl]piperazin-1-yl]-2-[[3-(2-aminoethyl)-1H-indol-5-yl]oxy]ethanoneIC5010000.0 [1]
(1R,9S,13S)-1,13-Dimethyl-10-(2-morpholin-4-ylethyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
5-[4-(1-Butyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-2-methoxy-benzoic acidIC5010000.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-1-benzotellurophene-2-carboxamideKi500.0 [1]
(1R,9S,13S)-10-[2-(Dimethylamino)ethyl]-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
1'-Benzylspiro[3,4-dihydrothiochromene-2,4'-piperidine] 1,1-dioxideKi10000.0 [1]
(1R,9S,13S)-10-[2-(Diethylamino)ethyl]-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
1'-Benzylspiro[3,4-dihydrothiochromene-2,4'-piperidine] 1-oxideKi10000.0 [1]
(1R,9S,13S)-10-[2-(Cyclohexylamino)ethyl]-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
(1R,9S,13S)-10-[2-(Azepan-1-yl)ethyl]-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
(1R,9S,13S)-1,13-Dimethyl-10-(2-pyrrolidin-1-ylethyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olKi10000.0 [1]
(7S)-19-Methoxy-5-methyl-2,5-diazatetracyclo[13.4.0.02,7.08,13]nonadeca-1(15),8,10,12,16,18-hexaeneKi60.0 [1]
(7R)-19-Methoxy-5-methyl-2,5-diazatetracyclo[13.4.0.02,7.08,13]nonadeca-1(15),8,10,12,16,18-hexaeneKi43.0 [1]
(1S,7Ar)-hexahydro-1H-pyrrolizin-1-ylmethyl 1H-indazole-3-carboxylateIC5010000.0 [1]
[(1R,8S)-2,3,5,6,7,8-Hexahydro-1H-pyrrolizin-1-yl]methyl 1-methylindazole-3-carboxylateIC5010000.0 [1]
1-[4-(Acetylaminomethyl)benzyl]-4-(4-fluorophenyl)piperazineKi1000.0 [1]
N-[4-[4-(3-Chloro-2-methoxyphenyl)piperazin-1-yl]butyl]tricyclo[8.2.2.24,7]hexadeca-1(13),4,6,10(14),11,15-hexaene-5-carboxamideKi470.0 [1]
N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-12-oxatetracyclo[8.5.2.24,7.011,15]nonadeca-1(15),4,6,10,13,16,18-heptaene-13-carboxamideKi2700.0 [1]
N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]tricyclo[8.2.2.24,7]hexadeca-1(13),4,6,10(14),11,15-hexaene-5-carboxamideKi3500.0 [1]
N-[4-[4-(2,3-Difluorophenyl)piperazin-1-yl]butyl]tricyclo[8.2.2.24,7]hexadeca-1(13),4,6,10(14),11,15-hexaene-5-carboxamideKi1200.0 [1]
4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-thiazol-2-ylamineKi37.0 [1]
Methyl 2-[(4-ethoxycarbonylpiperidin-1-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylateKi170.0 [1]
Methyl 2-[(4-anilino-4-carbamoylpiperidin-1-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylateKi171.0 [1]
2-[(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylic acidKi1722.0 [1]
2-[(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxamideKi1722.0 [1]
Butyl 2-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylateKi92.6 [1]
Benzyl 2-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylateKi143.0 [1]
N-(3-Phenylpropyl)-2-[(3-phenylpropylamino)methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxamideKi27.6 [1]
8-[[8-(Hydroxymethyl)-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indol-2-yl]methyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-oneKi1722.0 [1]
4-(6-(18F)Fluoranylpyridin-2-yl)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]benzamideKi450.0 [1]
4-(6-(18F)Fluoranylpyridin-3-yl)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]benzamideKi760.0 [1]
3-[4-(1-Furan-3-ylmethyl-1H-indol-3-yl)-piperidin-1-ylmethyl]-benzoic acidIC5010000.0 [1]
1-[4-(Acetylaminomethyl)benzyl]-4-(4-chlorophenyl)piperazineKi1000.0 [1]
1-[4-(Acetylaminomethyl)benzyl]-4-(4-methoxyphenyl)piperazineKi1000.0 [1]
N,N-Dimethyl-2-[(Z)-(3-methylthieno[2,3-b]pyrrolizin-8-ylidene)amino]oxyethanamineIC503162.28 [1]
1-[4-(Acetylaminomethyl)phenethyl]-4-phenylpiperazineKi130.0 [1]
4-Amino-N-(1-azatricyclo[3.3.1.13,7]decan-4-yl)-5-chloro-2-methoxybenzamideIC5010000.0 [1]
(6S,7R)-6-Methyl-N,N-dipropyl-6,7,8,9-tetrahydrobenzo[g][1]benzofuran-7-amineKi70.0 [1]
Methyl 2-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-3,7-dihydro-2H-[1,4]dioxino[2,3-e]indole-8-carboxylateKi31.6 [1]
2-[1-[(4-Methylphenyl)methyl]piperidin-4-yl]-3,4-dihydro-2H-naphthalen-1-one;hydrateKi52.0 [1]
2-Hydroxybutanedioic acid;1'-(naphthalen-2-ylmethyl)spiro[3,4-dihydronaphthalene-2,4'-piperidine]-1-oneKi1969.0 [1]
2-Hydroxybutanedioic acid;1'-[[4-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydronaphthalene-2,4'-piperidine]-1-oneKi6336.0 [1]
Items per page: 1 - 10 of 100
⟨⟩

References

This online tool may be cited as follows

MLA

"Quest Database™ Serotonin 2 (5-HT2) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/serotonin-2-5-ht2-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Serotonin 2 (5-HT2) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-2-5-ht2-receptor-inhibitors-ic50-ki.
BibTeXEndNoteRefMan
Location: Home / Datasets / Serotonin 2 (5-HT2) receptor Inhibitors (IC50, Ki)
AboutPrivacyTerms of UseTerms of SalesDistributors
Copyright © 2024 AAT Bioquest, Inc. All Rights Reserved.