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Serotonin 2a (5-HT2a) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ClozapineIC5012.0 [1]
ClozapineKi6.3 [1], 9.1 [2]
KetanserinIC5014.0 [1]
AripiprazoleIC501100.0 [1], 2790.0 [2]
OlanzapineIC509.0 [1], 100.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 2a (5-HT2a) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/serotonin-2a-5-ht2a-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseSerotonin 2a (5-HT2a) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-2a-5-ht2a-receptor-inhibitors-ic50-ki.
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