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Serotonin 2b (5-HT2b) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
4-Iodo-2,5-dimethoxyphenylisopropylamineIC502.5 [1], 3.2 [2], 3.5 [3], 4.0 [4]
4-Iodo-2,5-dimethoxyphenylisopropylamineKi1.6 [1], 2.0 [2], 42.7 [3]
SerotoninKi12.0 [1], 13.0 [2], 13.49 [3]
1-(3-Chlorophenyl)piperazineKi10.0 [1], 24.0 [2], 32.0 [3]
6-Chloro-5-methyl-1-((2-(2-methylpyrid-3-yloxy)pyrid-5-yl)carbamoyl)indolineKi100.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 2b (5-HT2b) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/serotonin-2b-5-ht2b-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseSerotonin 2b (5-HT2b) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-2b-5-ht2b-receptor-inhibitors-ic50-ki.
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