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Serotonin 3 (5-HT3) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
m-ChlorophenylbiguanideKi17.0 [1], 18.0 [2]
1-(3-Chlorophenyl)guanidineKi32.0 [1], 35.0 [2]
QuipazineIC500.45 [1]
QuipazineKi1.8 [1], 2.0 [2]
1-PhenylbiguanideKi1200.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 3 (5-HT3) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.7 Dec2025https://www.aatbio.com/data-sets/serotonin-3-5-ht3-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 7). Quest DatabaseSerotonin 3 (5-HT3) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-3-5-ht3-receptor-inhibitors-ic50-ki.
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