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Serotonin 3a (5-HT3a) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
BemesetronIC5010.0 [1]
BemesetronKi3.9 [1]
OndansetronIC500.09 [1]
OndansetronKi2.8 [1], 3.4 [2], 16.0 [3], 16.2 [4]
TropisetronKi2.7 [1], 2.82 [2], 5.3 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 3a (5-HT3a) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.22 Dec2025https://www.aatbio.com/data-sets/serotonin-3a-5-ht3a-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 22). Quest DatabaseSerotonin 3a (5-HT3a) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-3a-5-ht3a-receptor-inhibitors-ic50-ki.
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