Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| (1-(2-(Methylsulfonylamino)ethyl)-4-piperidinyl)methyl 1-methyl-1H-indole-3-carboxylate | IC50 | 0.21 [1] | |
| Piboserod | IC50 | 0.63 [1] | |
| Piboserod | Ki | 0.25 [1] | |
| Tegaserod | Ki | 3.98 [1], 31.0 [2] | |
| 2-Methoxy-4-amino-5-chlorobenzoic acid 2-(4-phenylpiperazino)ethyl ester | Ki | 12.5 [1], 14.3 [2], 23.0 [3], 32.0 [4], 55.0 [5] | |
MLA | "Quest Database™ Serotonin 4 (5-HT4) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/serotonin-4-5-ht4-receptor-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Serotonin 4 (5-HT4) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-4-5-ht4-receptor-inhibitors-ic50-ki. | |
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