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Serotonin 4 (5-HT4) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
(1-(2-(Methylsulfonylamino)ethyl)-4-piperidinyl)methyl 1-methyl-1H-indole-3-carboxylateIC500.21 [1]
PiboserodIC500.63 [1]
PiboserodKi0.25 [1]
TegaserodKi3.98 [1], 31.0 [2]
2-Methoxy-4-amino-5-chlorobenzoic acid 2-(4-phenylpiperazino)ethyl esterKi12.5 [1], 14.3 [2], 23.0 [3], 32.0 [4], 55.0 [5]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 4 (5-HT4) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/serotonin-4-5-ht4-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseSerotonin 4 (5-HT4) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-4-5-ht4-receptor-inhibitors-ic50-ki.
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