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Serotonin 5a (5-HT5a) receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
SerotoninIC5079.0 [1], 184.0 [2]
SerotoninKi110.0 [1], 126.0 [2], 130.0 [3], 170.0 [4], 250.0 [5]
ErgotamineKi14.0 [1], 16.0 [2], 22.0 [3], 40.0 [4]
8-OH-DpatKi1000.0 [1], 2500.0 [2]
MethiothepinKi1.0 [1], 100.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseSerotonin 5a (5-HT5a) receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.6 Dec2025https://www.aatbio.com/data-sets/serotonin-5a-5-ht5a-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 6). Quest DatabaseSerotonin 5a (5-HT5a) receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serotonin-5a-5-ht5a-receptor-inhibitors-ic50-ki.
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