SHC-transforming protein 1 Inhibitors (IC50, Ki)

Name: SHC-transforming protein 1 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	248000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-ethylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	19000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-propylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	25700.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-prop-2-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	26600.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-butylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	8900.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-but-3-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	6000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-benzylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	18900.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-but-2-ynylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	83000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(3-methylbutyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	17000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(4-fluorobutyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	40000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(4,4,4-trifluorobutyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	23000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(2-methoxyethyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	56000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(4-methylpentyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	29000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-pentylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	10000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-pent-4-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	16000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-pent-2-ynylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	17000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(2-ethoxyethyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	33000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(2-ethylsulfanylethyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	34000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-hexylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	20000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-hex-5-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	14000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-(4-cyanobutyl)amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	44000.0 ^[1]
	[4-[(2S)-2-[Acetyl(prop-2-enyl)amino]-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-[[(2S)-3-hydroxy-1-oxo-1-(prop-2-enylamino)propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	41000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-[[(2S)-3-hydroxy-1-oxo-1-(prop-2-enylamino)propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	189000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-[[(2S)-3-hydroxy-1-oxo-1-(prop-2-enylamino)propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-prop-2-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	48000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-[[(2S)-1-(but-3-enylamino)-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	165000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-4-methyl-1-oxo-1-(prop-2-enylamino)pentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	91000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-[[(2S)-3-hydroxy-1-oxo-1-(prop-2-enylamino)propan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-prop-2-enylamino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	353000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-4-methyl-1-oxo-1-(prop-2-enylamino)pentan-2-yl]-prop-2-enylamino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	81000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-4-methyl-1-oxo-1-(prop-2-enylamino)pentan-2-yl]amino]-2-oxoethyl]-prop-2-enylamino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	47000.0 ^[1]
	[4-[(2S)-2-[Acetyl(prop-2-enyl)amino]-3-[[(2S)-5-amino-1-[[2-[[(2S)-4-methyl-1-oxo-1-(prop-2-enylamino)pentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	450000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[[(2S)-1-(but-3-enylamino)-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	84000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[but-3-enyl-[(2S)-1-[[(2S)-1-(but-3-enylamino)-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	89000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[but-3-enyl-[2-[[(2S)-1-[[(2S)-1-(but-3-enylamino)-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	8000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[[2-[but-3-enyl-[(2S)-1-(but-3-enylamino)-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	84000.0 ^[1]
	[4-[(2S)-2-Acetamido-3-[[(2S)-5-amino-1-[but-3-enyl-[2-[[(2S)-1-(but-3-enylamino)-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1,5-dioxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate	IC50	14000.0 ^[1]

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References

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MLA	"Quest Database™ SHC-transforming protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/shc-transforming-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ SHC-transforming protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/shc-transforming-protein-1-inhibitors-ic50-ki.
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SHC-transforming protein 1 Inhibitors (IC50, Ki)

References

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