Short transient receptor potential channel 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	7-Bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide	IC50	25000.0 [1]
	3,4-Dihydro-1H-isoquinolin-2-yl-[2-(4-methoxyanilino)-1,3-thiazol-4-yl]methanone	IC50	1260.0 [1]
	4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide	IC50	39810.72 [1]
	(4-Methylpiperidino)[2-(4-toluidino)-1,3-thiazol-4-yl]methanone	IC50	630.0 [1]
	[2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2S,3S)-2,3-dimethylpiperidin-1-yl]methanone	IC50	100.0 [1]
	4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrile	IC50	10000.0 [1]
	{2-[(4-Methoxyphenyl)amino]-1,3-thiazol-4-yl}(4-methylpiperidin-1-yl)methanone	IC50	800.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone	IC50	500.0 [1]
	[2-(4-Chloroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone	IC50	800.0 [1]
	[2-(2-Chloroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone	IC50	6300.0 [1]
	[2-(4-Chloro-2-fluoroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone	IC50	1600.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone	IC50	400.0 [1]
	[2-(4-Methylanilino)-1,3-thiazol-4-yl]-(2-methylpiperidin-1-yl)methanone	IC50	800.0 [1]
	[2-(4-Methylanilino)-1,3-thiazol-4-yl]-(2-phenylpiperidin-1-yl)methanone	IC50	12600.0 [1]
	[2-(4-Methylanilino)-1,3-thiazol-4-yl]-(3-phenylpiperidin-1-yl)methanone	IC50	25000.0 [1]
	[2-(4-Methoxyanilino)-1,3-thiazol-4-yl]-(4-phenylpiperidin-1-yl)methanone	IC50	2500.0 [1]
	(4-Cyclohexylpiperidin-1-yl)-[2-(4-methylanilino)-1,3-thiazol-4-yl]methanone	IC50	6300.0 [1]
	(2,3-Dimethylpiperidin-1-yl)-[2-(4-methylanilino)-1,3-thiazol-4-yl]methanone	IC50	250.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone	IC50	80.0 [1]
	(2,3-Dimethylpiperidin-1-yl)-[2-[(6-fluoro-1,3-benzodioxol-5-yl)amino]-5-methyl-1,3-thiazol-4-yl]methanone	IC50	160.0 [1]
	[5-Chloro-2-[(6-fluoro-1,3-benzodioxol-5-yl)amino]-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone	IC50	32.0 [1]
	[2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone	IC50	250.0 [1]
	[2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2R,3R)-2,3-dimethylpiperidin-1-yl]methanone	IC50	1000.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)methanone	IC50	316.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]-(1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)methanone	IC50	316.0 [1]
	[2-(1,3-Benzodioxol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]-(5-methyl-7,8-dihydro-5H-1,6-naphthyridin-6-yl)methanone	IC50	10000.0 [1]
	[2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-(7,8-dihydro-5H-1,6-naphthyridin-6-yl)methanone	IC50	20000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 27 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Short transient receptor potential channel 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/short-transient-receptor-potential-channel-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Short transient receptor potential channel 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/short-transient-receptor-potential-channel-3-inhibitors-ic50-ki.
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