Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 6-(4-Chlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 15.7 [1], 168.0 [2] | |
| 5-[(4-Chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenoxy]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 584.0 [2] | |
| 5-[(4-Chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 1.91 [2] | |
| 6-(3-Chlorophenoxy)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 117.0 [2] | |
| 6-(4-Chlorophenyl)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.84 [1], 242.0 [2] | |
MLA | "Quest Database™ Short transient receptor potential channel 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 17 Dec. 2025, https://www.aatbio.com/data-sets/short-transient-receptor-potential-channel-5-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 17). Quest Database™ Short transient receptor potential channel 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/short-transient-receptor-potential-channel-5-inhibitors-ic50-ki. | |
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