Signal peptide peptidase-like 2A Inhibitors (IC50, Ki)

Name: Signal peptide peptidase-like 2A Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(2S)-2-Cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide	IC50	77.0 ^[1], 160.0 ^[2]
	LY-411575	IC50	10.0 ^[1]
	(Z-LL)2 ketone	IC50	6.0 ^[1]
	(2R)-2-Methyl-N'-(3-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	70.0 ^[1]
	(2R)-N'-(3,5-Difluorophenyl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	5.0 ^[1]
	(2R)-2-Methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-[2-(trifluoromethyl)phenyl]butanediamide	IC50	2850.0 ^[1]
	(2R)-2-Methyl-N'-(4-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	1390.0 ^[1]
	(2R)-N-[(6S)-5,11-Dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)-2-methylbutanediamide	IC50	870.0 ^[1]
	(2S)-2-Cyclopropyl-N-[(6S)-5,11-dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide	IC50	225.0 ^[1]
	(2R)-N'-(5-Fluoro-2-methylpyridin-3-yl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	44.0 ^[1]
	(2R)-2-Methyl-N'-(2-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	35.0 ^[1]
	(2R)-2-Methyl-N'-(2-methylpyridin-3-yl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide	IC50	1020.0 ^[1]
	(2R)-N'-(5-Fluoro-2-methylpyridin-3-yl)-N-[(6S)-10-fluoro-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-2-methylbutanediamide	IC50	76.0 ^[1]

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References

This online tool may be cited as follows

MLA	"Quest Database™ Signal peptide peptidase-like 2A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/signal-peptide-peptidase-like-2a-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Signal peptide peptidase-like 2A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/signal-peptide-peptidase-like-2a-inhibitors-ic50-ki.
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Signal peptide peptidase-like 2A Inhibitors (IC50, Ki)

References

This online tool may be cited as follows

MLA

APA