Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| (2S)-2-Cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide | IC50 | 77.0 [1], 160.0 [2] | |
| LY-411575 | IC50 | 10.0 [1] | |
| (Z-LL)2 ketone | IC50 | 6.0 [1] | |
| (2R)-2-Methyl-N'-(3-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide | IC50 | 70.0 [1] | |
| (2R)-N'-(3,5-Difluorophenyl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide | IC50 | 5.0 [1] | |
MLA | "Quest Database™ Signal peptide peptidase-like 2A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/signal-peptide-peptidase-like-2a-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ Signal peptide peptidase-like 2A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/signal-peptide-peptidase-like-2a-inhibitors-ic50-ki. | |
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