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Signal transducer and activator of transcription 5A Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
Azd-1480IC5025.0 [1], 41.0 [2]
SodiumIC509400.0 [1]
NF449 octasodium saltIC501400.0 [1]
6-(2,6-Dichlorophenyl)-2-[(4-Fluoro-3-Methylphenyl)amino]-8-Methylpyrido[2,3-D]pyrimidin-7(8h)-OneIC505.0 [1]
[4-[[[2-[6-(Phenylcarbamoyl)naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC504970.0 [1]
[4-[[[2-[4-[(4-Chlorophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC507400.0 [1]
[4-[[[2-[4-[(4-Bromophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC508600.0 [1]
[4-[[[2-[4-[(4-Fluorophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC508300.0 [1]
[4-[[[2-[4-[(3-Fluorophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC5011900.0 [1]
[4-[[[2-[4-[(3-Bromophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC5010500.0 [1]
[4-[[[2-[4-[(3-Chlorophenyl)carbamoyl]phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC509100.0 [1]
[4-[[[2-[4-(Phenylcarbamoyl)phenoxy]acetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC509700.0 [1]
[4-[[[2-[6-[(3-Bromophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC5010600.0 [1]
[4-[[[2-[6-[(4-Chlorophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC508900.0 [1]
[4-[[[2-[6-[(4-Bromophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC507600.0 [1]
[4-[[[2-[6-[(3-Fluorophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC508400.0 [1]
[4-[[[2-[6-[(3-Chlorophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC507300.0 [1]
[4-[[[2-[6-[(4-Fluorophenyl)carbamoyl]naphthalen-2-yl]oxyacetyl]amino]methyl]-2-phosphonooxyphenyl] dihydrogen phosphateIC507200.0 [1]
(16R,17S)-16,17-Dihydroxy-4,14,19-triazaheptacyclo[12.11.2.02,6.07,27.08,13.019,26.020,25]heptacosa-1,6,8,10,12,20,22,24,26-nonaen-3-oneIC50689.0 [1]
Hexasodium;8-[[3-[[3-[(4,6,8-trisulfonatonaphthalen-1-yl)carbamoyl]phenyl]carbamoylamino]benzoyl]amino]naphthalene-1,3,5-trisulfonate;hydrateIC508800.0 [1]
STAT5 InhibitorIC5047000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Signal transducer and activator of transcription 5A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/signal-transducer-and-activator-of-transcription-5a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Signal transducer and activator of transcription 5A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/signal-transducer-and-activator-of-transcription-5a-inhibitors-ic50-ki.
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