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Sodium channel alpha subunit Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
ChlorpromazineIC504300.0 [1]
HaloperidolIC507000.0 [1]
NifedipineIC5037000.0 [1]
AmiodaroneIC504800.0 [1]
ImipramineIC503600.0 [1]
AmitriptylineIC5020000.0 [1]
DiltiazemIC509000.0 [1]
PimozideIC5054.0 [1]
NitrendipineIC5036000.0 [1]
MexiletineIC5043000.0 [1]
DofetilideIC50300000.0 [1]
MibefradilIC50980.0 [1]
SertindoleIC502300.0 [1]
CibenzolineIC507800.0 [1]
TedisamilIC5020000.0 [1]
(18R)-13-Ethyl-8-methyl-8,15-diazahexacyclo[14.2.1.01,9.02,7.010,15.012,17]nonadeca-2,4,6-triene-14,18-diolIC508200.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Sodium channel alpha subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/sodium-channel-alpha-subunit-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Sodium channel alpha subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sodium-channel-alpha-subunit-inhibitors-ic50-ki.
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