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Sodium channel protein type III alpha subunit Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamideIC502450.0 [1], 11760.0 [2]
N-[[5-[1-(2-Imidazol-1-ylethyl)indazol-3-yl]-1,2,4-oxadiazol-3-yl]methyl]benzamideIC5022000.0 [1], 100000.0 [2]
N-[[5-[2-(2-Imidazol-1-ylethyl)indazol-3-yl]-1,2,4-oxadiazol-3-yl]methyl]-3-(trifluoromethoxy)benzamideIC504760.0 [1], 97000.0 [2], 100000.0 [3]
N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]-1,3,5-triazin-2-yl]amino]phenyl]acetamideIC50300.0 [1], 10000.0 [2]
2,2-Diphenyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamideIC5017.0 [1], 20.0 [2]
Tert-butyl 2-amino-4-[3-(1H-indole-2-carbonylamino)phenyl]imidazole-1-carboxylateIC5026000.0 [1], 30000.0 [2]
4-[(5-Chloro-1,3-thiazol-2-yl)sulfamoyl]-N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]benzamideIC5030.0 [1]
Tert-butyl 2-amino-4-[4-[[(2R)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylateIC5030000.0 [1]
Tert-butyl 4-[3-(furan-2-carbonylamino)phenyl]-2-(methylamino)imidazole-1-carboxylateIC5030000.0 [1]
Tert-butyl 2-amino-4-[4-(1H-indole-2-carbonylamino)phenyl]imidazole-1-carboxylateIC5022000.0 [1], 30000.0 [2]
N-[3-[2-Amino-1-(1H-pyrrole-2-carbonyl)imidazol-4-yl]phenyl]-1H-pyrrole-2-carboxamideIC5025000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[3-[[(2R)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylateIC5030000.0 [1]
Tert-butyl 2-amino-4-[3-(1H-indole-3-carbonylamino)phenyl]imidazole-1-carboxylateIC5027000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[3-(1H-pyrrole-3-carbonylamino)phenyl]imidazole-1-carboxylateIC5023000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[3-(1H-pyrrole-2-carbonylamino)phenyl]imidazole-1-carboxylateIC5025000.0 [1], 30000.0 [2]
Tert-butyl 4-[3-(1H-indole-2-carbonylamino)phenyl]-2-(methylamino)imidazole-1-carboxylateIC5030000.0 [1]
Tert-butyl 2-amino-4-[3-(1H-pyrrole-3-carbonylamino)phenyl]imidazole-1-carboxylate;hydrochlorideIC5012000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[4-(furan-2-carbonylamino)phenyl]imidazole-1-carboxylateIC5027000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[4-[[(2S)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylateIC5025000.0 [1], 30000.0 [2]
Tert-butyl 2-amino-4-[4-(1H-pyrrole-2-carbonylamino)phenyl]imidazole-1-carboxylateIC5030000.0 [1]
N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-3-carboxamideIC5012000.0 [1], 30000.0 [2]
N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-pyrrole-2-carboxamideIC5030000.0 [1]
N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-2-carboxamideIC5030000.0 [1]
N-[3-[2-(Methylamino)-1H-imidazol-5-yl]phenyl]-1H-indole-2-carboxamideIC5030000.0 [1]
N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-pyrrole-2-carboxamideIC5030000.0 [1]
N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-2-carboxamideIC5030000.0 [1]
(2R)-N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]pyrrolidine-2-carboxamideIC508000.0 [1], 30000.0 [2]
(2S)-N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]pyrrolidine-2-carboxamideIC5013000.0 [1], 30000.0 [2]
LidocaineIC5010500.0 [1]
TetrodotoxinIC5030.0 [1]
LamotrigineIC5017000.0 [1]
TetracaineIC50740.0 [1]
SenicapocIC501000.0 [1]
CID 46840946IC5010000.0 [1]
6-Amino-N-methyl-5-(2,3,5-trichlorophenyl)picolinamideIC5014000.0 [1]
1-[2-Methoxy-4-[3-(trifluoromethyl)phenyl]phenyl]-2-oxo-N-pyrimidin-2-ylquinoline-6-sulfonamideIC5042500.0 [1]
CID 118734430IC5020.3 [1]
N-[6-Amino-5-[2-(trifluoromethoxy)phenyl]pyridin-2-yl]-3-methyl-1,2-oxazole-4-carboxamideIC5010000.0 [1]
4-[4-Chloro-2-[2-(1-ethylazetidin-3-yl)pyrazol-3-yl]phenoxy]-3-cyano-N-(1,3-thiazol-4-yl)benzenesulfonamideIC5010000.0 [1]
5-Chloro-2-fluoro-4-[2-pyridazin-4-yl-4-(trifluoromethyl)phenoxy]-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamideIC5010000.0 [1]
4-[2-(2-Amino-3H-benzimidazol-5-yl)-4-chlorophenoxy]-2,5-difluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC509330.0 [1]
4-[4-Chloro-2-(2-methylpyrazol-3-yl)phenoxy]-3-fluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC50292.0 [1]
4-[4-Chloro-2-(2-methylpyrazol-3-yl)phenoxy]-3-cyano-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC503000.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1H-indole-2-carboxamideIC5030000.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-4,5-dibromo-1H-pyrrole-2-carboxamideIC5026000.0 [1]
N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-4,5-dibromo-1H-pyrrole-2-carboxamideIC5018000.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-4-bromo-1H-pyrrole-2-carboxamideIC5026000.0 [1]
4-[2-Methoxy-4-(trifluoromethyl)phenyl]-N-(1,3-thiazol-2-yl)quinazoline-7-sulfonamideIC5021000.0 [1]
N-[6-Amino-5-(2,3,5-trichlorophenyl)pyridin-2-yl]acetamideIC503500.0 [1]
3-Cyano-4-[2-[2-[(2-piperidin-4-ylethylamino)methyl]pyridin-4-yl]-4-[3-(trifluoromethyl)phenyl]phenoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC506438.0 [1]
1-[1-(2-Fluorophenyl)indazol-4-yl]-3-[2-[(3S)-3-fluoropyrrolidin-1-yl]-2-oxoethyl]imidazolidin-2-oneIC507100.0 [1]
1-[5-Fluoro-2-methoxy-4-[3-(trifluoromethyl)phenyl]phenyl]-N-(1,2-oxazol-3-yl)isoquinoline-6-sulfonamideIC506900.0 [1]
(3Ar,6aS)-5-[1-(2-fluorophenyl)indazol-4-yl]-2-(3-hydroxy-3-methylbutanoyl)-3,3a,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-4-oneIC5020000.0 [1]
1-[2-[5-Fluoro-1-(2-fluorophenyl)indazol-3-yl]oxyethyl]imidazolidin-2-oneIC503400.0 [1]
4-[(3S)-3-[(3R)-3-(3,5-Dichlorophenyl)pyrrolidin-1-yl]-2-oxopyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)benzenesulfonamideIC502000.0 [1]
6-Amino-N-methyl-5-(2,3,5-trichlorophenyl)pyridine-3-carboxamideIC506900.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1-methylpyrrole-2-carboxamideIC5024000.0 [1]
N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-1H-pyrrole-2-carboxamideIC5028000.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]furan-2-carboxamideIC5027000.0 [1]
Tert-butyl (2S)-2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]carbamoyl]pyrrolidine-1-carboxylateIC5030000.0 [1]
(6S)-6-N-(1H-Pyrrol-2-ylmethyl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamineIC5025000.0 [1]
N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-1H-indole-2-carboxamideIC5016000.0 [1]
Tert-butyl (2S)-2-[(2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methylcarbamoyl]pyrrolidine-1-carboxylateIC5026000.0 [1]
N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1H-pyrrole-2-carboxamideIC5030000.0 [1]
N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-4-bromo-1H-pyrrole-2-carboxamideIC5020000.0 [1]
2-Fluoro-N-(1,3-thiazol-2-yl)-4-[(3S)-3-[5-(trifluoromethyl)pyridin-2-yl]oxypyrrolidin-1-yl]sulfonylbenzenesulfonamideIC50851.0 [1]
2-Fluoro-N-(1,3-thiazol-2-yl)-4-[4-[6-(trifluoromethyl)pyridin-2-yl]piperidin-1-yl]sulfonylbenzenesulfonamideIC501640.0 [1]
2-Fluoro-4-(3-phenoxyazetidin-1-yl)sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamideIC50959.0 [1]
2-Fluoro-N-(1,2,4-thiadiazol-5-yl)-4-[4-[2-(trifluoromethyl)pyrimidin-4-yl]piperidine-1-carbonyl]benzenesulfonamideIC506675.0 [1]
4-[[3-Chloro-4-(trifluoromethoxy)phenyl]methoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC5022.0 [1]
4-[(3S)-3-(2,6-Dichlorophenoxy)pyrrolidin-1-yl]sulfonyl-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamideIC50945.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(1,2,4-thiadiazol-5-ylsulfamoyl)benzamideIC5013.0 [1]
4-N-(1,3-Thiazol-2-yl)-1-N-[[4-(trifluoromethyl)phenyl]methyl]benzene-1,4-disulfonamideIC50160.0 [1]
4-[3-Chloro-4-(trifluoromethoxy)phenoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC50296.0 [1]
2-Fluoro-4-[2-(3-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamideIC501830.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-[(5-fluoropyrimidin-2-yl)sulfamoyl]benzamideIC50993.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyrimidin-5-ylsulfamoyl)benzamideIC503000.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyrimidin-2-ylsulfamoyl)benzamideIC50374.0 [1]
2-Fluoro-N-(1,2,4-thiadiazol-5-yl)-4-[4-[5-[2-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl]piperidine-1-carbonyl]benzenesulfonamideIC501955.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-N-methyl-4-(1,2,4-thiadiazol-5-ylsulfamoyl)benzamideIC50522.0 [1]
N-(1,3-Thiazol-2-yl)-4-[5-[[4-(trifluoromethyl)phenyl]methyl]-1H-1,2,4-triazol-3-yl]benzenesulfonamideIC50124.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyridazin-3-ylsulfamoyl)benzamideIC501793.0 [1]
2-Fluoro-4-[(2R)-2-[(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)methyl]pyrrolidin-1-yl]sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamideIC503000.0 [1]
4-[[1-[3-Chloro-4-(trifluoromethoxy)benzoyl]azetidin-3-yl]oxymethyl]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamideIC50237.0 [1]
2-Phenyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamideIC503790.0 [1]
1-[2-(4-Fluorophenoxy)acetyl]-N-(1,3-thiazol-2-yl)-2,3-dihydroindole-5-sulfonamideIC502506.0 [1]
4-[5-[(3,4-Dichlorophenyl)methyl]-1H-1,2,4-triazol-3-yl]-N-(1,3-thiazol-2-yl)benzenesulfonamideIC5045.0 [1]
N-(1,3-Thiazol-2-yl)-4-[2-[4-(trifluoromethyl)phenyl]ethylsulfonyl]benzenesulfonamideIC50155.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-4-(1,3-thiazol-2-ylsulfamoyl)benzamideIC5020.0 [1]
N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(1,3-thiazol-2-ylsulfamoyl)benzamideIC5011.0 [1]
4-(1,3-Thiazol-2-ylsulfamoyl)-N-[[4-(trifluoromethyl)phenyl]methyl]benzamideIC50147.0 [1]
1-[2-(4-Fluorophenoxy)acetyl]-N-(1,2,4-thiadiazol-5-yl)-2,3-dihydroindole-5-sulfonamideIC501273.0 [1]
(2S)-N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]pyrrolidine-2-carboxamideIC5030000.0 [1]
(2S)-N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]pyrrolidine-2-carboxamideIC5030000.0 [1]
N-Benzyl-4-(1,3-thiazol-2-ylsulfamoyl)benzamideIC504450.0 [1]
4-(1,3-Thiazol-2-ylsulfamoyl)-N-[[4-(trifluoromethoxy)phenyl]methyl]benzamideIC50197.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Sodium channel protein type III alpha subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 7 May. 2024, https://www.aatbio.com/data-sets/sodium-channel-protein-type-iii-alpha-subunit-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 7). Quest Database™ Sodium channel protein type III alpha subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sodium-channel-protein-type-iii-alpha-subunit-inhibitors-ic50-ki.
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